SCHEMBL8084928

SCHEMBL8084928

CC1Oc2ccc([N+](=O)[O-])cc2C(Oc2ccc(O)nn2)C1(C)O

nearest known ligand 0.37

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.37
HIF1A Q16665 1/20 0.31
HSP90AA1 P07900 1/20 0.31
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7334818 0.82 AKR1B1 (0.35) AKR1B1HIF1AHSP90AA1ALDH1A1
SCHEMBL7331033 0.76 ABCC9 (0.35) AKR1B1HIF1AHSP90AA1ALDH1A1
SCHEMBL7321412 0.75 ABCC9 (0.39) AKR1B1HIF1AHSP90AA1ALDH1A1
SCHEMBL7330893 0.74 TLR3 (0.40) AKR1B1HIF1AHSP90AA1ALDH1A1
SCHEMBL7326918 0.72 AKR1B1 (0.35) AKR1B1ALDH1A1
SCHEMBL9377381 0.65 KDM4E (0.36) AKR1B1ALDH1A1
SCHEMBL7332017 0.65 ALDH1A1 (0.30) ALDH1A1
SCHEMBL7323754 0.65 ABCC9 (0.39) AKR1B1HIF1AHSP90AA1ALDH1A1
SCHEMBL7332446 0.64 MAPT (0.33) AKR1B1HIF1AALDH1A1
SCHEMBL8085025 0.64 AKR1B1 (0.33) AKR1B1HIF1AHSP90AA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
EP-0340718-B1 Chroman derivatives MERCK PATENT GMBH (DE) 1994-07-20 EP disclosed
US-5013853-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-05-07 US disclosed
EP-0340718-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1989-11-08 EP disclosed