SCHEMBL8085141

SCHEMBL8085141

CC(=O)Oc1cccn(C2=CC(C)(C)Oc3ccc([N+](=O)[O-])cc32)c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.44
POLB P06746 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HSP90AA1 P07900 1/20 0.36
CCR6 P51684 1/20 0.36
KDM4E B2RXH2 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADORA2A P29274 1/20 0.35
TYMS P04818 1/20 0.34
ALDH1A1 P00352 1/20 0.33
MAPT P10636 2/20 0.33
LMNA P02545 1/20 0.33
RAB9A P51151 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MALT1 Q9UDY8 1/20 0.32
CA9 Q16790 3/20 0.32
CA12 O43570 2/20 0.32
CA1 P00915 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8088445 0.89 ADORA3 (0.41) RECQLTDP1KDM4EHTTSMN1; SMN2
SCHEMBL8088352 0.86 KDM4E (0.37) RECQLTDP1HSP90AA1KDM4EHTT
SCHEMBL10697020 0.85 ALDH1A1 (0.36) RECQLTDP1HTTSMN1; SMN2ALDH1A1
SCHEMBL8084289 0.83 CFTR (0.41) RECQLTDP1KDM4EHTTSMN1; SMN2
SCHEMBL8090699 0.83 ALDH1A1 (0.37) POLBTDP1KDM4EHTTALDH1A1
SCHEMBL8085305 0.83 ALDH1A1 (0.36) TDP1HTTALDH1A1MALT1CA9
SCHEMBL8077039 0.83 ALDH1A1 (0.36) TDP1HTTALDH1A1MALT1CA9
SCHEMBL7274143 0.82 PDE4A (0.42) KDM4EADORA3ADORA2ATYMSMALT1
SCHEMBL8088675 0.82 RECQL (0.44) RECQLPOLBTDP1HSP90AA1CCR6
SCHEMBL7292380 0.80 CCNC (0.32) KDM4EADORA3ADORA2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed