SCHEMBL8077334

SCHEMBL8077334

CC1=C(n2cccc([N+](=O)[O-])c2=O)c2cc([N+](=O)[O-])ccc2OC1(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
POLB P06746 1/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
CTDSP1 Q9GZU7 1/20 0.35
MALT1 Q9UDY8 1/20 0.35
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34
GABRA3 P34903 1/20 0.34
CYP3A4 P08684 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PTPRC P08575 3/20 0.33
S100A4 P26447 2/20 0.33
CASP1 P29466 1/20 0.33
CASP3 P42574 1/20 0.33
CASP4 P49662 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8084426 0.88 ALDH1A1 (0.36) ALDH1A1MEN1KMT2AMALT1CYP3A4
SCHEMBL8077303 0.88 ALDH1A1 (0.36) ALDH1A1MEN1KMT2AMALT1GABRA1
SCHEMBL8076907 0.88 TDP1 (0.37) ALDH1A1MEN1KMT2AMALT1CYP3A4
SCHEMBL8076882 0.87 ABCC9 (0.37) POLBMEN1KMT2AMALT1TDP1
SCHEMBL8085347 0.86 ADORA3 (0.36) ALDH1A1MEN1KMT2ACYP3A4TDP1
SCHEMBL8076960 0.86 MEN1 (0.37) ALDH1A1POLBMEN1KMT2ACTDSP1
SCHEMBL8090492 0.85 KDM4E (0.36) ALDH1A1POLBMEN1KMT2AMALT1
SCHEMBL8085346 0.84 ALDH1A1 (0.38) ALDH1A1POLBMEN1KMT2AMALT1
SCHEMBL8088847 0.84 MYC (0.38) ALDH1A1POLBMEN1KMT2ACYP3A4
SCHEMBL8088675 0.84 RECQL (0.44) ALDH1A1POLBMEN1KMT2AMALT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
US-5013853-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-05-07 US disclosed