SCHEMBL8086539

SCHEMBL8086539

CC(C)(C)c1ccccc1S(=O)(=O)NC(Cc1ccccc1)C(=O)O

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.67
MAPT P10636 1/20 0.67
MMP2 P08253 9/20 0.59
MMP9 P14780 8/20 0.59
ADAMTS4 O75173 1/20 0.59
POLB P06746 2/20 0.58
HTT P42858 1/20 0.56
ADAMTS5 Q9UNA0 1/20 0.53
MMP1 P03956 1/20 0.53
MMP3 P08254 1/20 0.53
MMP7 P09237 1/20 0.53
MMP13 P45452 1/20 0.53
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5502394 0.83 POLB (0.66) ALDH1A1MAPTMMP2MMP9ADAMTS4
SCHEMBL6670956 0.83 POLB (0.66) ALDH1A1MAPTMMP2MMP9ADAMTS4
SCHEMBL11589175 0.83 MMP9 (0.46) ALDH1A1MAPTMMP2MMP9ADAMTS4
SCHEMBL6916882 0.82 MMP2 (0.63) ALDH1A1MAPTMMP2MMP9ADAMTS4
SCHEMBL11952564 0.81 MMP2 (0.62) ALDH1A1MAPTMMP2MMP9ADAMTS4
SCHEMBL11950557 0.81 MMP2 (0.62) ALDH1A1MAPTMMP2MMP9ADAMTS4
SCHEMBL6522675 0.81 MMP2 (0.66) ALDH1A1MAPTMMP2MMP9ADAMTS4
SCHEMBL31086837 0.80 ALDH1A1 (1.00) ALDH1A1MAPTMMP2MMP9ADAMTS4
SCHEMBL698062 0.79 MMP2 (0.63) ALDH1A1MAPTMMP2MMP9ADAMTS4
SCHEMBL698061 0.79 MMP2 (0.63) ALDH1A1MAPTMMP2MMP9ADAMTS4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0817795-B1 NOVEL 4-SUBSTITUTED-3-PEPTIDYL-AZETIDIN-2-ONE DERIVATIVES USEFUL AS CYSTEINE PROTEINASE INHIBITOR NAEJA PHARMACEUTICAL INC (CA) 2000-11-15 EP claimed
US-5986108-A ENZYME INHIBITORS SYNPHAR LABORATORIES, INC. (CA) 1999-11-16 US claimed