SCHEMBL8089404

SCHEMBL8089404

CCCCc1nc2cc[nH]c(=O)c2n1Cc1ccc(NC(=O)c2ccccc2C(=O)O)cc1

nearest known ligand 0.74

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 4/20 0.74
AGTR1 P30556 3/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8081250 0.86 AGTR2 (0.72) AGTR2AGTR1
SCHEMBL8092218 0.86 AGTR2 (0.60) AGTR2AGTR1
SCHEMBL8094878 0.85 AGTR2 (0.58) AGTR2AGTR1
SCHEMBL8089484 0.85 AGTR2 (1.00) AGTR2AGTR1
SCHEMBL8089288 0.84 AGTR1 (0.60) AGTR2AGTR1
SCHEMBL8081240 0.82 AGTR2 (0.73) AGTR2AGTR1
SCHEMBL8089320 0.79 AGTR2 (0.82) AGTR2AGTR1
SCHEMBL8094963 0.79 AGTR2 (0.68) AGTR2AGTR1
SCHEMBL8089261 0.79 AGTR2 (0.68) AGTR2AGTR1
SCHEMBL9031922 0.77 AGTR1 (0.61) AGTR2AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6037349-A HAVING ANTAGONISTIC PROPERTIES TOWARDS ANGIOTENSIN II CAN BE USED FOR THE TREATMENT OF HYPERTENSION, ALDOSTERONISM AND CARDIAC INSUFFICIENCY MERCK PATENT GMBH (DE) 2000-03-14 US disclosed
EP-0505893-A1 Imidazopyridines MERCK PATENT GmbH (DE) 1992-09-30 EP disclosed