SCHEMBL8089518

SCHEMBL8089518

CO[C@H]1C[C@]2(C)C(=C(F)F)CC[C@H]2[C@@H]2CCc3cc(OC4CCCCO4)ccc3[C@H]21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.51
AKR1C3 P42330 3/20 0.44
MAPK1 P28482 2/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ESR1 P03372 4/20 0.39
ESR2 Q92731 1/20 0.39
MAPT P10636 3/20 0.36
LMNA P02545 2/20 0.36
HSD17B1 P14061 1/20 0.36
RECQL P46063 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
STS P08842 3/20 0.34
ABCC4 O15439 1/20 0.34
CYP2C9 P11712 1/20 0.34
ABCC1 P33527 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8088710 0.87 AKR1C3 (0.56) HSD11B1AKR1C3MAPK1TSHRHSD17B10
SCHEMBL7827752 0.84 HSD11B1 (0.69) HSD11B1MAPK1HSD17B10ESR1ESR2
SCHEMBL7830895 0.84 HSD11B1 (0.69) HSD11B1MAPK1HSD17B10ESR1ESR2
SCHEMBL8088769 0.80 AKR1C3 (0.59) AKR1C3MAPK1TSHRHSD17B10ESR1
SCHEMBL1657336 0.75 HSD11B1 (0.67) HSD11B1MAPK1HSD17B10ESR1ESR2
SCHEMBL8089481 0.73 HSD11B1 (0.52) HSD11B1MAPK1HSD17B10ESR1MAPT
SCHEMBL8089786 0.72 HSD11B1 (0.45) HSD11B1
SCHEMBL1657830 0.72 HSD11B1 (0.69) HSD11B1HSD17B10ESR1ESR2MAPT
SCHEMBL7830892 0.72 HSD11B1 (0.69) HSD11B1HSD17B10ESR1ESR2MAPT
SCHEMBL7830967 0.70 ALDH1A1 (0.46) HSD11B1LMNAKDM4EALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6136800-A STEROIDS SCHERING AKTIENGESELLSCHAFT (DE) 2000-10-24 US disclosed
US-6018062-A SUCH AS 17-DIFLUOROMETHYLENE-ESTRA-1,3,5(10)-TRIEN-3-OL; USE AS ANTIOXIDANTS AND VASCULOPROTECTIVE AGENTS AS THEY CAUSE VASODILATOR NITROGEN OXIDE RELEASE AND PREVENT OXIDATION OF LDL CHOLESTEROL SCHERING AKTIENGESELLSCHAFT (DE) 2000-01-25 US disclosed