SCHEMBL8088710

SCHEMBL8088710

CO[C@H]1C[C@]2(C)C(=O)CC[C@H]2[C@@H]2CCc3cc(OC4CCCCO4)ccc3[C@H]21

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.56
HSD17B10 Q99714 2/20 0.51
TSHR P16473 1/20 0.51
MAPK1 P28482 1/20 0.51
HSD11B1 P28845 1/20 0.51
MAPT P10636 3/20 0.48
LMNA P02545 2/20 0.48
HSD17B1 P14061 2/20 0.48
RECQL P46063 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
STS P08842 6/20 0.44
ESR1 P03372 3/20 0.43
ESR2 Q92731 3/20 0.43
KDM4E B2RXH2 2/20 0.43
ABCC4 O15439 1/20 0.43
CYP2C9 P11712 1/20 0.43
ABCC1 P33527 1/20 0.43
SLCO1B1 Q9Y6L6 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8089518 0.87 HSD11B1 (0.51) AKR1C3HSD17B10TSHRMAPK1HSD11B1
SCHEMBL1657830 0.83 HSD11B1 (0.69) HSD17B10HSD11B1MAPTLMNAHSD17B1
SCHEMBL7830892 0.83 HSD11B1 (0.69) HSD17B10HSD11B1MAPTLMNAHSD17B1
SCHEMBL8216067 0.80 STS (0.67) AKR1C3HSD17B10TSHRMAPK1MAPT
SCHEMBL6866735 0.80 STS (0.67) AKR1C3HSD17B10TSHRMAPK1MAPT
SCHEMBL5681977 0.78 AKR1C3 (0.79) AKR1C3HSD17B10TSHRMAPK1MAPT
SCHEMBL11101736 0.73 HSD17B1 (0.67) AKR1C3HSD17B10TSHRMAPK1MAPT
SCHEMBL15999637 0.72 AKR1C3 (1.00) AKR1C3HSD17B10TSHRMAPK1MAPT
SCHEMBL9634078 0.72 LMNA (0.66) AKR1C3HSD17B10TSHRMAPK1MAPT
SCHEMBL9746964 0.72 HSD17B1 (0.66) AKR1C3HSD17B10TSHRMAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6136800-A STEROIDS SCHERING AKTIENGESELLSCHAFT (DE) 2000-10-24 US disclosed
US-6018062-A SUCH AS 17-DIFLUOROMETHYLENE-ESTRA-1,3,5(10)-TRIEN-3-OL; USE AS ANTIOXIDANTS AND VASCULOPROTECTIVE AGENTS AS THEY CAUSE VASODILATOR NITROGEN OXIDE RELEASE AND PREVENT OXIDATION OF LDL CHOLESTEROL SCHERING AKTIENGESELLSCHAFT (DE) 2000-01-25 US disclosed