SCHEMBL8089807

SCHEMBL8089807

CC(=O)OC1C(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C(=O)N1N

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSK P43235 9/20 0.54
CTSS P25774 8/20 0.54
CTSL P07711 7/20 0.54
ALDH1A1 P00352 1/20 0.50
ALOX15 P16050 1/20 0.50
CTSB P07858 9/20 0.48
TACR1 P25103 2/20 0.47
ELANE P08246 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7441597 1.00 CTSK (0.54) CTSKCTSSCTSLALDH1A1ALOX15
SCHEMBL8085377 0.90 CTSK (0.55) CTSKCTSSCTSLCTSB
SCHEMBL8086169 0.89 GNPAT (0.44) CTSKCTSSCTSLALDH1A1TACR1
SCHEMBL7436065 0.88 CTSK (0.45) CTSKCTSSCTSLCTSBELANE
SCHEMBL7444607 0.88 CTSK (0.54) CTSKCTSSCTSLALDH1A1ALOX15
SCHEMBL8086238 0.87 CTSK (0.55) CTSKCTSSCTSLALDH1A1ALOX15
SCHEMBL7442716 0.86 CTSK (0.55) CTSKCTSSCTSLALDH1A1ALOX15
SCHEMBL7441709 0.85 CTSL (0.56) CTSKCTSSCTSLALDH1A1ALOX15
SCHEMBL7451264 0.84 FAAH (0.43) ALDH1A1
SCHEMBL7438536 0.82 NOS2 (0.48) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0817795-B1 NOVEL 4-SUBSTITUTED-3-PEPTIDYL-AZETIDIN-2-ONE DERIVATIVES USEFUL AS CYSTEINE PROTEINASE INHIBITOR NAEJA PHARMACEUTICAL INC (CA) 2000-11-15 EP disclosed