SCHEMBL8090145

SCHEMBL8090145

N=c1ccn(CCC[C@H](NC(=O)C2(C(=O)NCCc3ccccc3)CCCC2)OBO)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 2/20 0.35
CHRM3 P20309 2/20 0.35
MMP8 P22894 2/20 0.35
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
CHRM1 P11229 1/20 0.33
TACR1 P25103 1/20 0.33
TACR3 P29371 1/20 0.33
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
FPR3 P25089 1/20 0.32
FPR2 P25090 1/20 0.32
PSEN1 P49768 4/20 0.32
PSEN2 P49810 4/20 0.32
APH1B Q8WW43 4/20 0.32
NCSTN Q92542 4/20 0.32
APH1A Q96BI3 4/20 0.32
PSENEN Q9NZ42 4/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8090141 0.94 CHRM5 (0.36) CHRM5CHRM3MMP8CYP3A4CYP2C19
SCHEMBL8095467 0.84 CYP3A4 (0.38) MMP8CYP3A4CYP2C19TACR1TACR3
SCHEMBL8090113 0.84 CYP2C19 (0.38) CHRM5CHRM3MMP8CYP3A4CYP2C19
SCHEMBL8095269 0.83 MMP1 (0.38) MMP8CYP3A4CYP2C19EPHX1
Hydrochloric Acid SCHEMBL7432966 0.83 F2 (0.37) CHRM5CHRM3MMP8CYP3A4CYP2C19
SCHEMBL8090189 0.82 MMP8 (0.37) MMP8CYP3A4CYP2C19TACR1TACR3
SCHEMBL8098091 0.79 MMP8 (0.43) MMP8CYP2C19ALDH1A1NPC1EPHX2
SCHEMBL8095221 0.79 MMP8 (0.41) MMP8CYP2C19EPHX2CNR1
SCHEMBL8090112 0.77 CYP2C19 (0.39) MMP8CYP3A4CYP2C19TACR1TACR3
SCHEMBL8095466 0.77 CYP2C19 (0.39) MMP8CYP3A4CYP2C19TACR1TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0792883-B1 Novel derivates of boronic acid, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2000-12-20 EP disclosed
EP-0792883-A1 Novel derivates of boronic acid, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1997-09-03 EP disclosed