SCHEMBL8095466

SCHEMBL8095466

NCCCC(NC(=O)C1(C(=O)NCCc2ccccc2)CCCC1)OBOC(CCCN)NC(=O)C1(C(=O)NCCc2ccccc2)CCCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 3/20 0.39
CYP3A4 P08684 2/20 0.39
MMP8 P22894 2/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
KDM4E B2RXH2 1/20 0.37
CYP1A2 P05177 1/20 0.37
TACR1 P25103 1/20 0.37
TACR3 P29371 1/20 0.37
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
EPHX1 P07099 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
MMP1 P03956 1/20 0.35
MMP3 P08254 1/20 0.35
MMP9 P14780 1/20 0.35
F2 P00734 3/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8095266 0.97 MMP1 (0.39) CYP2C19CYP3A4MMP8MEN1KMT2A
SCHEMBL8098087 0.95 MMP8 (0.44) CYP2C19MMP8KMT2ANPC1ALDH1A1
SCHEMBL8095467 0.93 CYP3A4 (0.38) CYP2C19CYP3A4MMP8MEN1KMT2A
SCHEMBL8090127 0.92 KDM4E (0.36) CYP2C19KDM4ECYP1A2NR1H2NR1H3
SCHEMBL8095269 0.90 MMP1 (0.38) CYP2C19CYP3A4MMP8EPHX1MMP1
SCHEMBL8090112 0.90 CYP2C19 (0.39) CYP2C19CYP3A4MMP8MEN1KMT2A
SCHEMBL8095182 0.90 MMP8 (0.40) CYP2C19MMP8CYP1A2EPHX1MMP1
SCHEMBL8091668 0.89 MMP8 (0.39) MMP8EPHX1MMP1ALDH1A1
SCHEMBL8091392 0.89 CYP2A6 (0.38) CYP3A4MEN1KMT2AEPHX1NPC1
SCHEMBL8090174 0.89 F2 (0.39) CYP2C19CYP3A4MMP8MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0792883-B1 Novel derivates of boronic acid, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2000-12-20 EP disclosed
EP-0792883-A1 Novel derivates of boronic acid, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1997-09-03 EP disclosed