SCHEMBL8090448

SCHEMBL8090448

Cc1ccc(F)c([Si](C)(C)C)c1C#N

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.35
GFER P55789 1/20 0.35
KDM4E B2RXH2 4/20 0.35
ALDH1A1 P00352 3/20 0.35
MAPT P10636 2/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
HSD17B10 Q99714 1/20 0.35
APOBEC3G Q9HC16 1/20 0.35
LMNA P02545 4/20 0.35
POLB P06746 2/20 0.34
RAB9A P51151 2/20 0.34
XBP1 P17861 1/20 0.34
MAPK1 P28482 1/20 0.34
ATM Q13315 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CYP1A2 P05177 3/20 0.33
CYP2C19 P33261 2/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10120481 0.75 CYP1A2 (0.37) GAAGFERKDM4EALDH1A1MAPT
SCHEMBL13082493 0.75 CYP1A2 (0.37) GAAGFERKDM4EALDH1A1MAPT
SCHEMBL6734851 0.74 ACHE (0.35)
SCHEMBL8112763 0.72 ALDH1A1 (0.36) GAAGFERKDM4EALDH1A1MAPT
SCHEMBL16136624 0.71 TRPV4 (0.37) GAAGFERKDM4EALDH1A1MAPT
SCHEMBL17192918 0.71 TRPV4 (0.37) GAAGFERKDM4EALDH1A1MAPT
SCHEMBL7975208 0.71 CYP1A2 (0.46) GAAKDM4EALDH1A1MAPTHPGD
SCHEMBL31050110 0.71 CYP1A2 (0.46) GAAKDM4EALDH1A1MAPTHPGD
SCHEMBL14051608 0.70 CYP1A2 (0.39) KDM4EALDH1A1MAPTHPGDALOX15
SCHEMBL13748182 0.69 AKR1B1 (0.33) GAAGFERKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1221407-A Aminoisoquinolines and aminothienopyridine derivatives and their use as anti-inflammatory agents ASTRA PHARMA PROD (GB) 1999-06-30 CN claimed
EP-0892784-A1 AMINOISOQUINOLINES AND AMINOTHIENOPYRIDINE DERIVATIVES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS Astra Pharmaceuticals Limited (GB) 1999-01-27 EP claimed
WO-1997038977-A1 AMINOISOQUINOLINES AND AMINOTHIENOPYRIDINE DERIVATIVES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS ASTRA PHARMACEUTICALS LTD. (GB) 1997-10-23 WO claimed
US-6063789-A Aminoisoquinolines and aminotheinopyridine derivatives and their use as anti-inflammatory agents ASTRA PHARMACEUTICALS, LTD. (GB) 2000-05-16 US disclosed
CN-1221407-A Aminoisoquinolines and aminothienopyridine derivatives and their use as anti-inflammatory agents ASTRA PHARMA PROD (GB) 1999-06-30 CN disclosed
EP-0892784-A1 AMINOISOQUINOLINES AND AMINOTHIENOPYRIDINE DERIVATIVES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS Astra Pharmaceuticals Limited (GB) 1999-01-27 EP disclosed
WO-1997038977-A1 AMINOISOQUINOLINES AND AMINOTHIENOPYRIDINE DERIVATIVES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS ASTRA PHARMACEUTICALS LTD. (GB) 1997-10-23 WO disclosed