Aspartame

Aspartame

SCHEMBL8091203

COC(=O)[C@H](Cc1ccccc1)NC(=O)C(N)CC(=O)O

nearest known ligand 0.64

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.64
THRB P10828 1/20 0.64
CYP2C9 P11712 1/20 0.64
CYP2C19 P33261 1/20 0.64
HSD17B10 Q99714 1/20 0.64
OPRK1 P41145 1/20 0.58
ATM Q13315 2/20 0.58
POLB P06746 1/20 0.55
BIRC2 Q13490 1/20 0.54
LMNA P02545 1/20 0.53
GLA P06280 1/20 0.53
TSHR P16473 1/20 0.53
ANPEP P15144 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Aspartame SCHEMBL19283498 1.00 ALDH1A1 (0.64) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
Aspartame SCHEMBL10625481 1.00 ALDH1A1 (0.64) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
Aspartame SCHEMBL28591 1.00 ALDH1A1 (0.64) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
Aspartame SCHEMBL900809 1.00 ALDH1A1 (0.64) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
Aspartame SCHEMBL216238 1.00 ALDH1A1 (0.64) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
Aspartame SCHEMBL3637 1.00 ALDH1A1 (0.64) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
Aspartame SCHEMBL10635593 1.00 ALDH1A1 (0.64) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
Aspartame SCHEMBL11085391 1.00 ALDH1A1 (0.64) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
Aspartame SCHEMBL8761655 1.00 ALDH1A1 (0.64) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
Aspartame SCHEMBL3636 1.00 ALDH1A1 (0.64) ALDH1A1THRBCYP2C9CYP2C19HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 50 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109996778-B Taste modifying aldehydes 高砂香料工业株式会社 2022-12-13 CN claimed
EP-0581032-B1 Method for production of alpha-L-aspartyl-L-phenylalanine methyl ester hydrochloride AJINOMOTO KK (JP) 1997-06-11 EP claimed
EP-0523813-B1 Method for crystallizing alpha-L-aspartyl-L-phenylalanine methyl ester HOLLAND SWEETENER CO (NL) 1996-11-27 EP claimed
US-5304671-A Solid-liquid separation of suspension; no desalting; precipitation of acid salt; neutralization; hydrolysis AJINOMOTO CO., INC. (JP) 1994-04-19 US claimed
EP-0581032-A1 Method for production of alpha-L-aspartyl-L-phenylalanine methyl ester hydrochloride Ajinomoto Co., Inc. (JP) 1994-02-02 EP claimed
EP-0523813-A1 Method for crystallizing alpha-L-aspartyl-L-phenylalanine methyl ester HOLLAND SWEETENER COMPANY V.O.F. (NL) 1993-01-20 EP claimed
EP-0302478-B1 METHOD FOR PURIFYING A DIPEPTIDE ESTER Tosoh Corporation (JP) 1992-05-06 EP claimed
US-4944852-A Method for purifying a dipeptide ester TOSOH CORPORATION (JP) 1990-07-31 US claimed
US-4831180-A GRANULATING WET CRYSTALS, DRYING TOYO SODA MANUFACTURING COMPANY, LTD. (JP) 1989-05-16 US claimed
US-4824994-A Method for production of N-protected-alpha-L-aspartyl-L-phenylalanine methyl ester AJINOMOTO CO., INC. (JP) 1989-04-25 US claimed
US-4810818-A MULTISTAGE DRYING TOYO SODA MANUFACTURING CO., LTD (JP) 1989-03-07 US claimed
EP-0302478-A1 Method for purifying a dipeptide ester Tosoh Corporation (JP) 1989-02-08 EP claimed
EP-0227007-A2 N-(4-benzyl-L-alpha-aspartyl)-L-phenylalanine methyl ester, its process of preparation and its use HOECHST AKTIENGESELLSCHAFT (DE) 1987-07-01 EP claimed
US-4638081-A Process for preparing α-aspartyl-L-phenylalanine methyl ester DE-BI DERIVATI BIOLOGICI INTERNATIONAL SPA (IT) 1987-01-20 US claimed
JP-5117246-A None JP disclosed
JP-1040498-A None JP disclosed
JP-63159355-A None JP disclosed
US-4549987-A DEFORMYLATION AND SEPARATION OF N-FORMYL-L-A-ASPARTYL-L-PHENYLALANINE METHYL ESTER FARMITALIA CARLO ERBA S.P.A. (IT) 1985-10-29 US disclosed
US-4549987-A DEFORMYLATION AND SEPARATION OF N-FORMYL-L-A-ASPARTYL-L-PHENYLALANINE METHYL ESTER FARMITALIA CARLO ERBA S.P.A. (IT) 1985-10-29 US disclosed
EP-0132856-A2 Process for preparing alpha-L-aspartyl-L-phenylalanine methyl ester DE-BI DERIVATI BIOLOGICI INTERNATIONAL S.p.A. (IT) 1985-02-13 EP disclosed