SCHEMBL8091378

SCHEMBL8091378

O=C(Nc1ccc(Cl)cc1)NS(=O)(=O)Cc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 5/20 0.57
NPC1 O15118 2/20 0.57
RAB9A P51151 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
ALDH1A1 P00352 3/20 0.50
ACP1 P24666 2/20 0.49
MET P08581 1/20 0.48
IDH1 O75874 2/20 0.48
CASR P41180 1/20 0.48
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
MEN1 O00255 1/20 0.48
CA12 O43570 1/20 0.48
KMT2A Q03164 1/20 0.48
CA9 Q16790 1/20 0.48
MMP1 P03956 1/20 0.47
MMP2 P08253 1/20 0.47
MMP9 P14780 1/20 0.47
MMP8 P22894 1/20 0.47
MMP13 P45452 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6464498 0.89 ACP1 (0.61) SMN1; SMN2ACP1METCA1CA2
SCHEMBL6469561 0.88 CNR1 (0.50) CNR1NPC1RAB9AALDH1A1MET
SCHEMBL6463105 0.87 CA1 (0.57) ACP1METCA1CA2CA12
SCHEMBL8094923 0.86 CNR1 (0.55) CNR1NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL6468349 0.84 PGR (0.62) SMN1; SMN2METCA1CA2CA12
SCHEMBL6467730 0.82 ACP1 (0.51) NPC1RAB9AALDH1A1ACP1MET
SCHEMBL6466509 0.82 MET (0.61) NPC1RAB9ASMN1; SMN2ALDH1A1MET
SCHEMBL15145832 0.81 ALDH1A1 (0.56) CNR1NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL29400026 0.81 NAMPT (0.58) ALDH1A1MEN1KMT2A
SCHEMBL23747462 0.80 NAMPT (0.73) CNR1NPC1RAB9ASMN1; SMN2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0467621-B1 N-phenyl-N'-alkylsulfonylureas, process for their preparation and antitumor compositions containing them LILLY CO ELI (US) 1994-06-15 EP claimed
EP-0467621-A1 N-phenyl-N'-alkylsulfonylureas, process for their preparation and antitumor compositions containing them ELI LILLY AND COMPANY (US) 1992-01-22 EP claimed
US-6147115-A SULFONYLUREIDO-4-HALOBENZENE DERIVATIVES; ANTICARCINOGENIC AGENTS ELI LILLY AND COMPANY (US) 2000-11-14 US disclosed
EP-0467621-B1 N-phenyl-N'-alkylsulfonylureas, process for their preparation and antitumor compositions containing them LILLY CO ELI (US) 1994-06-15 EP disclosed
US-5216026-A Administering to the mammal N-1-butanesulfonamide derivatives and salts ELI LILLY AND COMPANY (US) 1993-06-01 US disclosed
EP-0467621-A1 N-phenyl-N'-alkylsulfonylureas, process for their preparation and antitumor compositions containing them ELI LILLY AND COMPANY (US) 1992-01-22 EP disclosed