SCHEMBL8091387

SCHEMBL8091387

CC(C)S(=O)(=O)NC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1

nearest known ligand 0.68

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.68
CA1 P00915 7/20 0.60
CA2 P00918 7/20 0.60
CA7 P43166 7/20 0.60
CA9 Q16790 7/20 0.60
PDK1 Q15118 1/20 0.58
TRPV1 Q8NER1 7/20 0.54
CNR2 P34972 1/20 0.54
CASR P41180 1/20 0.52
HDAC1 Q13547 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8083234 0.84 EPHX1 (0.62) CA1CA2CA9
SCHEMBL29364392 0.82 KDR (1.00) KDRCA1CA2CA7CA9
SCHEMBL118026 0.82 KDR (1.00) KDRCA1CA2CA7CA9
SCHEMBL12154419 0.81 KDR (0.75) KDRCA1CA2CA7CA9
SCHEMBL19605881 0.80 KDR (0.78) KDRCA1CA2CA7CA9
SCHEMBL8094995 0.80 LMNA (0.61) CA2
SCHEMBL8091384 0.80 KDR (0.64) KDRCA1CA2CA7CA9
SCHEMBL12413876 0.79 KDR (0.82) KDRCA1CA2CA7CA9
SCHEMBL8097749 0.79 LMNA (0.60) CA2
SCHEMBL10819632 0.78 PDK1 (0.76) KDRCA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6147115-A SULFONYLUREIDO-4-HALOBENZENE DERIVATIVES; ANTICARCINOGENIC AGENTS ELI LILLY AND COMPANY (US) 2000-11-14 US claimed
EP-0467621-B1 N-phenyl-N'-alkylsulfonylureas, process for their preparation and antitumor compositions containing them LILLY CO ELI (US) 1994-06-15 EP claimed
EP-0467621-A1 N-phenyl-N'-alkylsulfonylureas, process for their preparation and antitumor compositions containing them ELI LILLY AND COMPANY (US) 1992-01-22 EP claimed
US-6147115-A SULFONYLUREIDO-4-HALOBENZENE DERIVATIVES; ANTICARCINOGENIC AGENTS ELI LILLY AND COMPANY (US) 2000-11-14 US disclosed
EP-0467621-B1 N-phenyl-N'-alkylsulfonylureas, process for their preparation and antitumor compositions containing them LILLY CO ELI (US) 1994-06-15 EP disclosed
US-5216026-A Administering to the mammal N-1-butanesulfonamide derivatives and salts ELI LILLY AND COMPANY (US) 1993-06-01 US disclosed
EP-0467621-A1 N-phenyl-N'-alkylsulfonylureas, process for their preparation and antitumor compositions containing them ELI LILLY AND COMPANY (US) 1992-01-22 EP disclosed