SCHEMBL8091459

SCHEMBL8091459

CCC(Cc1ccccc1)NCCC(C)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.54
ADORA3 P0DMS8 2/20 0.54
SLC6A2 P23975 2/20 0.54
SLC6A4 P31645 2/20 0.54
ADRA1A P35348 2/20 0.54
OPRM1 P35372 2/20 0.54
DRD3 P35462 2/20 0.54
SLC6A3 Q01959 2/20 0.54
KCNH2 Q12809 2/20 0.54
ADRB2 P07550 1/20 0.54
ADRB1 P08588 1/20 0.54
DRD2 P14416 1/20 0.54
ADRA2B P18089 1/20 0.54
ADRA2C P18825 1/20 0.54
CNR1 P21554 1/20 0.54
HTR2A P28223 1/20 0.54
MC4R P32245 1/20 0.54
HRH1 P35367 1/20 0.54
SCN1A P35498 1/20 0.54
OPRK1 P41145 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8976808 0.80 SIGMAR1 (0.65) SLC6A4SIGMAR1MEN1KMT2A
SCHEMBL9150896 0.78 SIGMAR1 (0.62) SIGMAR1MEN1KMT2A
SCHEMBL22957649 0.78 HTR1A (0.53) HTR1AADORA3SLC6A2SLC6A4ADRA1A
SCHEMBL14064842 0.76 CYP3A4 (0.55) HTR1AADORA3SLC6A2SLC6A4ADRA1A
SCHEMBL22558398 0.76 SLC6A4 (0.62) SLC6A4SIGMAR1
SCHEMBL15131060 0.74 CYP3A4 (0.75) HTR1AADORA3SLC6A2SLC6A4ADRA1A
SCHEMBL8096613 0.74 SIGMAR1 (0.77) SIGMAR1MEN1KMT2A
SCHEMBL19750615 0.73 HTR1A (0.51) HTR1AADORA3SLC6A2SLC6A4ADRA1A
SCHEMBL21243263 0.73 SIGMAR1 (0.53) SLC6A2SLC6A4SLC6A3SIGMAR1
SCHEMBL7152487 0.73 ADRB2 (0.61) ADRB2ADRB1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057371-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, GASTROINTESTINAL DISORDERS, DRUG ABUSE, ANGINA, MIGRAINE, HYPERTENSION AND DEPRESSION VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-05-02 US disclosed
EP-0591426-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-04-13 EP disclosed
WO-1993000313-A2 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1993-01-07 WO disclosed