SCHEMBL8091536

SCHEMBL8091536

O=S(=O)(OC(c1ccccc1)c1nnn[nH]1)C(F)(F)F

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
IDO1 P14902 2/20 0.31
TDO2 P48775 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29856072 0.79 IDO1 (0.40) ALDH1A1MAPTMAPK1HTTKMT2A
Ammonia Solution, Strong SCHEMBL29119872 0.78 IDO1 (0.39) ALDH1A1MAPTMAPK1HTTKMT2A
SCHEMBL5450128 0.74 KMT2A (0.33) MAPK1HTTKMT2A
SCHEMBL7445813 0.70 ADRA2A (0.38)
SCHEMBL11639976 0.68 ALDH1A1 (0.43) ALDH1A1MAPTKMT2ANPSR1
SCHEMBL9090435 0.68 CES2 (0.33) ALDH1A1MAPK1HTTKMT2A
SCHEMBL7510243 0.67 KMT2A (0.44) ALDH1A1KMT2A
SCHEMBL11531757 0.67 KMT2A (0.35) ALDH1A1KMT2A
SCHEMBL1273034 0.66 NPSR1 (0.39) ALDH1A1MAPTMAPK1HTTKMT2A
SCHEMBL21831821 0.66 IDO1 (0.45) KMT2AIDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0829480-B1 Tetrazolyl-substituted quinuclidines as substance P antagonists PFIZER (US) 2000-12-20 EP disclosed
US-5939434-A Tetrazolyl-substituted quinuclidines as substance P antagonists PFIZER PHARMACEUTICALS INC. (JP) 1999-08-17 US disclosed
EP-0829480-A2 Tetrazolyl-substituted quinuclidines as substance P antagonists PFIZER INC. (US) 1998-03-18 EP disclosed