SCHEMBL8092078

SCHEMBL8092078

CS(=O)(=O)Nc1cc(CCC(=O)O)c([N+](=O)[O-])cc1Oc1ccc(Cl)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.48
PTGS2 P35354 2/20 0.48
CCR2 P41597 1/20 0.45
FFAR1 O14842 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
PTGDR Q13258 5/20 0.41
PTGDR2 Q9Y5Y4 5/20 0.41
MAPT P10636 5/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
POLB P06746 1/20 0.41
PKM P14618 1/20 0.41
CHRM1 P11229 1/20 0.40
CYP19A1 P11511 2/20 0.39
GAA P10253 1/20 0.39
S1PR4 O95977 1/20 0.39
CPT1A P50416 1/20 0.38
CPT1B Q92523 1/20 0.38
LMNA P02545 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8476355 0.92 PTGS1 (0.48) PTGS1PTGS2CCR2TDP1MAPT
SCHEMBL8525177 0.87 PTGS1 (0.50) PTGS1PTGS2CCR2TDP1PTGDR
SCHEMBL8524014 0.85 PTGS1 (0.46) PTGS1PTGS2CCR2TDP1PTGDR
SCHEMBL8092076 0.80 PTGS1 (0.47) PTGS1PTGS2CCR2TDP1PTGDR
SCHEMBL7160901 0.80 FFAR1 (0.60) PTGS1PTGS2CCR2FFAR1PTGDR
SCHEMBL8476353 0.77 TDP1 (0.46) PTGS1PTGS2CCR2TDP1MAPT
SCHEMBL8524150 0.72 PTGS1 (0.54) PTGS1PTGS2CCR2PTGDRPTGDR2
SCHEMBL8481656 0.72 PTGS1 (0.51) PTGS1PTGS2CCR2FFAR1TDP1
SCHEMBL8101582 0.71 PTGS1 (0.50) PTGS1PTGS2CCR2PTGDRPTGDR2
SCHEMBL2394825 0.71 PTGDR2 (0.53) PTGS1PTGS2FFAR1TDP1PTGDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848703-B1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 2000-09-27 EP disclosed