SCHEMBL8092090

SCHEMBL8092090

Cc1cc(Cl)ccc1Sc1cc(S(N)(=O)=O)ccc1NS(C)(=O)=O

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.44
PTGS1 P23219 1/20 0.44
CCR2 P41597 5/20 0.41
CA2 P00918 9/20 0.40
CA1 P00915 7/20 0.40
CA9 Q16790 7/20 0.40
CA12 O43570 4/20 0.39
CA3 P07451 1/20 0.37
CA4 P22748 1/20 0.37
CA6 P23280 1/20 0.37
CA5A P35218 1/20 0.37
CA7 P43166 1/20 0.37
CA13 Q8N1Q1 1/20 0.37
CA14 Q9ULX7 1/20 0.37
CA5B Q9Y2D0 1/20 0.37
APP P05067 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4575696 0.89 PTGS1 (0.56) PTGS2PTGS1CCR2CA2CA1
SCHEMBL8479236 0.88 PTGS1 (0.44) PTGS2PTGS1CCR2CA2CA1
SCHEMBL8099531 0.88 CA1 (0.41) PTGS2CA2CA1CA9CA12
SCHEMBL8098762 0.86 PTGS1 (0.45) PTGS2PTGS1CCR2CA2CA1
SCHEMBL8100934 0.84 CA2 (0.44) PTGS2PTGS1CCR2CA2CA1
SCHEMBL8091883 0.83 PTGS1 (0.44) PTGS2PTGS1CA2CA1CA9
SCHEMBL8107618 0.81 NR3C1 (0.42) PTGS2PTGS1CA2CA1CA9
SCHEMBL8101100 0.80 CA2 (0.44) PTGS2PTGS1CA2CA1CA9
SCHEMBL8101110 0.80 CA2 (0.44) PTGS2PTGS1CA2CA1CA9
SCHEMBL8098886 0.78 CA2 (0.46) CA2CA1CA9CA12CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848703-B1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 2000-09-27 EP disclosed
US-6004948-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS; SIDE EFFECT REDUCTION NYCOMED AUSTRIA GMBH (AT) 1999-12-21 US disclosed