SCHEMBL8093075

SCHEMBL8093075

CC(C)(C)OC(=O)NC(Cc1ccc(OCc2ccccc2)cc1)C(O)C(F)(F)C(=O)NC(COCc1ccccc1)COCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 2/20 0.48
REN P00797 3/20 0.47
BCL2 P10415 1/20 0.47
PTPN1 P18031 3/20 0.46
PPARG P37231 1/20 0.45
CTSS P25774 1/20 0.44
MAOB P27338 1/20 0.43
KLK5 Q9Y337 2/20 0.43
YAP1 P46937 2/20 0.42
ATM Q13315 1/20 0.42
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42
LTA4H P09960 1/20 0.41
HDAC8 Q9BY41 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8945614 0.91 REN (0.47) PPARARENBCL2PTPN1PPARG
SCHEMBL8945512 0.91 REN (0.47) PPARARENBCL2PTPN1PPARG
SCHEMBL7331235 0.87 BCL2 (0.55) PPARARENBCL2PTPN1CTSS
SCHEMBL7422374 0.86 BCL2 (0.49) RENBCL2PTPN1KLK5ATM
SCHEMBL7417399 0.86 REN (0.47) PPARARENBCL2PTPN1KLK5
SCHEMBL8945503 0.86 REN (0.49) RENBCL2PTPN1KLK5YAP1
SCHEMBL7418529 0.85 REN (0.47) PPARARENBCL2PTPN1KLK5
SCHEMBL7421310 0.84 REN (0.49) PPARARENBCL2PTPN1MAOB
SCHEMBL7427451 0.84 REN (0.46) RENBCL2PTPN1KLK5YAP1
SCHEMBL8736231 0.84 BCL2 (0.49) PPARARENBCL2PTPN1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114380-A ANTIVIRAL AGENT; ADMINISTERING TO TREAT HIV INFECTION; N-(4-(N-BENZYLOXYCARBONYL-L-VALYL)AMINO-2,2-DIFLUORO-1,3-DIOXO-5-(4-(2-N -MORPHOLYL)ETHYLOXY)PHENYL-PENTYL)-O-((2-PYRIDYL)METHYL)-D-VALINOL, FOR EXAMPLE MERRELL PHARMACEUTICALS INC. (US) 2000-09-05 US disclosed