SCHEMBL8093408

SCHEMBL8093408

CC1NCC(=O)N(CC(=O)N(c2ccccc2)C(C)C)c2ccccc21

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
CCKAR P32238 16/20 0.44
CCKBR P32239 14/20 0.44
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8795637 0.78 ALDH1A1 (0.66) ALDH1A1CCKARCCKBRLMNATP53
SCHEMBL8807834 0.73 CCKAR (0.58) ALDH1A1CCKARCCKBR
SCHEMBL6904258 0.72 ALDH1A1 (0.52) ALDH1A1CCKARCCKBRLMNATP53
SCHEMBL8089873 0.71 CCKAR (0.55) ALDH1A1CCKARCCKBR
SCHEMBL5100093 0.68 ALDH1A1 (0.52) ALDH1A1CCKARCCKBRLMNATP53
SCHEMBL8709141 0.67 ALDH1A1 (0.59) ALDH1A1CCKARCCKBRLMNATP53
SCHEMBL5103627 0.67 CCKAR (0.65) ALDH1A1CCKARCCKBR
SCHEMBL8805668 0.67 CCKAR (0.52) ALDH1A1CCKARCCKBR
SCHEMBL8803465 0.67 ALDH1A1 (0.50) ALDH1A1CCKARCCKBR
SCHEMBL8804010 0.67 CCKAR (0.61) ALDH1A1CCKARCCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096885-A EXHIBIT AGONIST ACTIVITY FOR CCK-A RECEPTORS THEREBY ENABLING THEM TO MODULATE THE HORMONES GASTRIN AND CHOLECYSTOKININ IN MAMMALS. GLAXO WELLCOME INC. (US) 2000-08-01 US disclosed
EP-0785944-A1 ACYL AMINO ACETAMIDE DERIVATIVES WITH AGONIST ACTIVITY FOR CCK-A RECEPTORS GLAXO WELLCOME INC. (US) 1997-07-30 EP disclosed
WO-1996011940-A1 ACYL AMINO ACETAMIDE DERIVATIVES WITH AGONIST ACTIVITY FOR CCK-A RECEPTORS GLAXO WELLCOME INC. (US) 1996-04-25 WO disclosed