SCHEMBL6904258

SCHEMBL6904258

CC(C)N(C(=O)CN1C(=O)[C]CC(C(N)=O)c2ccccc21)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
CCKAR P32238 15/20 0.44
CCKBR P32239 14/20 0.44
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8093477 0.75 ALDH1A1 (0.61) ALDH1A1CCKARCCKBRLMNATP53
SCHEMBL8093408 0.72 ALDH1A1 (0.55) ALDH1A1CCKARCCKBRLMNATP53
SCHEMBL7752992 0.71 CCKAR (0.65) ALDH1A1CCKARCCKBR
SCHEMBL8081898 0.69 ALDH1A1 (0.45) ALDH1A1CCKARCCKBRLMNATP53
SCHEMBL7550570 0.69 CCKAR (0.67) ALDH1A1CCKARCCKBR
SCHEMBL8807834 0.68 CCKAR (0.58) ALDH1A1CCKARCCKBR
SCHEMBL8795883 0.67 ALDH1A1 (0.58) ALDH1A1CCKARCCKBR
SCHEMBL17993540 0.66 ALDH1A1 (0.65) ALDH1A1CCKARCCKBRLMNATP53
SCHEMBL8795637 0.65 ALDH1A1 (0.66) ALDH1A1CCKARCCKBRLMNATP53
SCHEMBL8817635 0.65 CCKAR (0.78) ALDH1A1CCKARCCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040002495-A1 Lactam glycogen phosphorylase inhibitors and method of use BRISTOL-MYERS SQUIBB COMPANY 2004-01-01 US claimed
US-6096885-A EXHIBIT AGONIST ACTIVITY FOR CCK-A RECEPTORS THEREBY ENABLING THEM TO MODULATE THE HORMONES GASTRIN AND CHOLECYSTOKININ IN MAMMALS. GLAXO WELLCOME INC. (US) 2000-08-01 US disclosed
EP-0785944-A1 ACYL AMINO ACETAMIDE DERIVATIVES WITH AGONIST ACTIVITY FOR CCK-A RECEPTORS GLAXO WELLCOME INC. (US) 1997-07-30 EP disclosed
WO-1996011940-A1 ACYL AMINO ACETAMIDE DERIVATIVES WITH AGONIST ACTIVITY FOR CCK-A RECEPTORS GLAXO WELLCOME INC. (US) 1996-04-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040002495-A1 Lactam glycogen phosphorylase inhibitors and method of use PYGL, PYGM, GYS2 ALDH1A1 2992/4885CCKAR 1739/4885CCKBR 3021/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.