SCHEMBL8093430

SCHEMBL8093430

O=C(Nc1ccccc1)N[C@H]1CCCCNC1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.62
FPR2 P25090 2/20 0.58
KDM4E B2RXH2 1/20 0.57
RAB9A P51151 3/20 0.56
EPHX1 P07099 1/20 0.56
EPHX2 P34913 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
CHEK1 O14757 1/20 0.54
CCR2 P41597 8/20 0.54
NPC1 O15118 1/20 0.50
JAK3 P52333 1/20 0.49
FPR1 P21462 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21182827 0.90 EPHX2 (0.53) ALDH1A1FPR2KDM4ERAB9AEPHX1
SCHEMBL8381645 0.80 RAB9A (0.75) ALDH1A1KDM4ERAB9ACHEK1CCR2
SCHEMBL15087624 0.80 RAB9A (0.75) ALDH1A1KDM4ERAB9ACHEK1CCR2
SCHEMBL10593938 0.79 ALDH1A1 (0.56) ALDH1A1FPR2KDM4ERAB9ACHEK1
SCHEMBL8095765 0.78 ALDH1A1 (0.52) ALDH1A1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL319610 0.77 CCR2 (0.68) ALDH1A1KDM4ERAB9ACCR2NPC1
SCHEMBL3487757 0.77 CCR2 (0.68) ALDH1A1KDM4ERAB9ACCR2NPC1
SCHEMBL3241217 0.77 CCR2 (0.68) ALDH1A1KDM4ERAB9ACCR2NPC1
SCHEMBL23874550 0.76 CRBN (0.66) RAB9AEPHX1EPHX2SMN1; SMN2MEN1
SCHEMBL21182644 0.76 FPR2 (0.57) ALDH1A1FPR2RAB9AEPHX1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096885-A EXHIBIT AGONIST ACTIVITY FOR CCK-A RECEPTORS THEREBY ENABLING THEM TO MODULATE THE HORMONES GASTRIN AND CHOLECYSTOKININ IN MAMMALS. GLAXO WELLCOME INC. (US) 2000-08-01 US disclosed
EP-0785944-A1 ACYL AMINO ACETAMIDE DERIVATIVES WITH AGONIST ACTIVITY FOR CCK-A RECEPTORS GLAXO WELLCOME INC. (US) 1997-07-30 EP disclosed
WO-1996011940-A1 ACYL AMINO ACETAMIDE DERIVATIVES WITH AGONIST ACTIVITY FOR CCK-A RECEPTORS GLAXO WELLCOME INC. (US) 1996-04-25 WO disclosed