SCHEMBL8093477

SCHEMBL8093477

CC(C)N(C(=O)CN1C(=O)[C]C(C(N)=O)C(=O)c2ccccc21)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.61
CCKAR P32238 14/20 0.43
CCKBR P32239 12/20 0.43
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6904258 0.75 ALDH1A1 (0.52) ALDH1A1CCKARCCKBRLMNATP53
SCHEMBL8795883 0.73 ALDH1A1 (0.58) ALDH1A1CCKARCCKBR
SCHEMBL8796363 0.72 ALDH1A1 (0.62) ALDH1A1CCKARCCKBRLMNATP53
Bromide SCHEMBL8795194 0.71 ALDH1A1 (0.61) ALDH1A1CCKARCCKBR
SCHEMBL8794022 0.71 ALDH1A1 (0.60) ALDH1A1CCKARCCKBR
SCHEMBL8795637 0.70 ALDH1A1 (0.66) ALDH1A1CCKARCCKBRLMNATP53
SCHEMBL7752992 0.70 CCKAR (0.65) ALDH1A1CCKARCCKBR
Bromide SCHEMBL8795033 0.70 ALDH1A1 (0.59) ALDH1A1CCKARCCKBR
Bromide SCHEMBL8795037 0.70 ALDH1A1 (0.59) ALDH1A1CCKARCCKBR
SCHEMBL8703893 0.69 ALDH1A1 (0.57) ALDH1A1CCKARCCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096885-A EXHIBIT AGONIST ACTIVITY FOR CCK-A RECEPTORS THEREBY ENABLING THEM TO MODULATE THE HORMONES GASTRIN AND CHOLECYSTOKININ IN MAMMALS. GLAXO WELLCOME INC. (US) 2000-08-01 US disclosed
EP-0785944-A1 ACYL AMINO ACETAMIDE DERIVATIVES WITH AGONIST ACTIVITY FOR CCK-A RECEPTORS GLAXO WELLCOME INC. (US) 1997-07-30 EP disclosed
WO-1996011940-A1 ACYL AMINO ACETAMIDE DERIVATIVES WITH AGONIST ACTIVITY FOR CCK-A RECEPTORS GLAXO WELLCOME INC. (US) 1996-04-25 WO disclosed