SCHEMBL8093710

SCHEMBL8093710

N#Cc1cc(-c2ccc(S(N)(=O)=O)cc2)c(-c2ccc(F)cc2)nc1OCc1cccs1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 11/20 0.47
PTGS2 P35354 7/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
PTGS1 P23219 5/20 0.40
CNR2 P34972 1/20 0.40
KIT P10721 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8096151 0.91 PTGS2 (0.49) CNR1PTGS2PTGS1
SCHEMBL8086461 0.86 CNR1 (0.61) CNR1PTGS2CA12CA1CA2
SCHEMBL8093875 0.85 CNR1 (0.64) CNR1PTGS2CA12CA1CA2
SCHEMBL8101248 0.84 CNR1 (0.47) CNR1PTGS2CA12CA1CA2
SCHEMBL8094551 0.83 CNR1 (0.49) CNR1PTGS2CA12CA1CA2
SCHEMBL8086490 0.83 ALDH1A1 (0.42) CNR1PTGS2CA12CA1CA2
SCHEMBL8095797 0.82 CNR1 (0.69) CNR1PTGS2CA12CA1CA2
SCHEMBL8094678 0.81 SQOR (0.53) CNR1PTGS2CNR2
SCHEMBL8095521 0.81 CNR1 (0.52) CNR1PTGS2CA12CA1CA2
SCHEMBL8094547 0.81 PTGS2 (0.60) CNR1PTGS2CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed