SCHEMBL8096618

SCHEMBL8096618

CC[CH]C(NCCCCc1ccccc1)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 16/20 0.53
L3MBTL1 Q9Y468 1/20 0.49
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9150904 0.89 SIGMAR1 (0.49) SIGMAR1KCNH2
SCHEMBL9373860 0.88 SIGMAR1 (0.52) SIGMAR1L3MBTL1MEN1KMT2A
SCHEMBL8091279 0.84 SIGMAR1 (0.50) SIGMAR1MEN1KMT2AKCNH2
SCHEMBL9374331 0.81 SIGMAR1 (0.49) SIGMAR1MEN1KMT2AKCNH2
SCHEMBL8976810 0.80 SIGMAR1 (0.44) SIGMAR1MEN1KMT2AKCNH2
SCHEMBL8099628 0.76 EPHX2 (0.57) SIGMAR1L3MBTL1MEN1KMT2A
SCHEMBL15131171 0.76 SIGMAR1 (0.65) SIGMAR1L3MBTL1MEN1KMT2AKCNH2
SCHEMBL8091460 0.75 CYP3A4 (0.45) MEN1KMT2AKCNH2
SCHEMBL12312527 0.73 SIGMAR1 (0.71) SIGMAR1L3MBTL1KMT2A
SCHEMBL8092975 0.73 SIGMAR1 (0.62) SIGMAR1L3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057371-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, GASTROINTESTINAL DISORDERS, DRUG ABUSE, ANGINA, MIGRAINE, HYPERTENSION AND DEPRESSION VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-05-02 US disclosed
EP-0591426-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-04-13 EP disclosed
WO-1993000313-A2 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1993-01-07 WO disclosed