SCHEMBL8096671

SCHEMBL8096671

CCC(NCCCc1ccc2ccccc2c1)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 6/20 0.61
EPHX2 P34913 2/20 0.47
CYP1A2 P05177 2/20 0.46
BCHE P06276 3/20 0.45
CYP2A6 P11509 1/20 0.44
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
CASR P41180 1/20 0.41
KDM4A O75164 1/20 0.40
MC4R P32245 1/20 0.40
MC5R P33032 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8099628 0.79 EPHX2 (0.57) SIGMAR1EPHX2KDM4A
SCHEMBL8096670 0.76 SIGMAR1 (1.00) SIGMAR1
SCHEMBL8091056 0.75 SIGMAR1 (0.58) SIGMAR1CYP1A2BCHECASRMC4R
SCHEMBL12301554 0.74 SIGMAR1 (0.56) SIGMAR1CYP1A2BCHECYP2A6HDAC1
SCHEMBL20545401 0.74 ALDH1A1 (0.50) SIGMAR1EPHX2HDAC1
SCHEMBL9666471 0.74 SIGMAR1 (0.59) SIGMAR1CYP1A2CYP2A6HDAC1HDAC8
SCHEMBL24504966 0.72 SMN1; SMN2 (0.54) EPHX2HDAC1
SCHEMBL9373302 0.72 SIGMAR1 (0.68) SIGMAR1CYP1A2MC4RMC5R
SCHEMBL20908974 0.72 SMN1; SMN2 (0.54) EPHX2HDAC1
SCHEMBL15901399 0.72 EPHX2 (0.42) EPHX2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057371-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, GASTROINTESTINAL DISORDERS, DRUG ABUSE, ANGINA, MIGRAINE, HYPERTENSION AND DEPRESSION VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-05-02 US disclosed