SCHEMBL8097434

SCHEMBL8097434

CC(Cc1ccc(C#N)cc1)(NC(=O)[C@H]1CCCN(C(=O)c2cccc(Cl)c2)C1)c1cnc[nH]1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.48
FNTA P49354 1/20 0.48
FNTB P49356 1/20 0.48
PGGT1B P53609 1/20 0.48
ALDH1A1 P00352 1/20 0.47
RHOA P61586 12/20 0.42
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8088938 0.86 KDM4E (0.46) KCNH2FNTAFNTBPGGT1BALDH1A1
SCHEMBL8097852 0.86 KDM4E (0.46) KCNH2FNTAFNTBPGGT1BALDH1A1
SCHEMBL8088954 0.85 ATM (0.46) ALDH1A1MEN1KMT2A
SCHEMBL8103721 0.83 ITGB3 (0.39) KMT2A
SCHEMBL8088811 0.83 GPR119 (0.44) ALDH1A1MEN1KMT2A
SCHEMBL8097458 0.83 ALOX12 (0.36) ALDH1A1MEN1KMT2A
SCHEMBL8098292 0.83 ATM (0.38) ALDH1A1MEN1KMT2A
SCHEMBL8104346 0.83 HPGD (0.43) ALDH1A1RHOAKMT2A
SCHEMBL8095919 0.82 ALOX12 (0.40) KMT2A
SCHEMBL8088397 0.82 GAA (0.39) FNTAFNTBALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127366-A ANTICARCINOGENIC OR ANTITUMOR AGENTS MERCK & CO., INC. (US) 2000-10-03 US disclosed
EP-0862435-A4 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO INC (US) 1999-02-03 EP disclosed
US-5817678-A IMIDAZOLE-CONTAINING PIPERIDINE DERIVATIVES, PEPTIDEMIMETIC MERCK & CO., INC. (US) 1998-10-06 US disclosed
EP-0862435-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1998-09-09 EP disclosed
WO-1997018813-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1997-05-29 WO disclosed