SCHEMBL8088811

SCHEMBL8088811

CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NC(C)(Cc2ccc(C#N)cc2)c2cnc[nH]2)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 4/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
KMT2A Q03164 1/20 0.44
MMP13 P45452 1/20 0.37
ADAM17 P78536 1/20 0.37
PRMT5 O14744 1/20 0.37
ITGB1 P05556 1/20 0.37
ITGA4 P13612 1/20 0.37
GPBAR1 Q8TDU6 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
ERG P11308 1/20 0.36
CYP2C9 P11712 1/20 0.36
PARP1 P09874 2/20 0.36
PARP2 Q9UGN5 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
TSHR P16473 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8444117 0.87 GPR119 (0.42) GPR119CYP11B1CYP11B2JAK2JAK1
SCHEMBL8096857 0.87 GPR119 (0.42) GPR119CYP11B1CYP11B2JAK2JAK1
SCHEMBL8097494 0.87 GPR119 (0.42) GPR119CYP11B1CYP11B2JAK2JAK1
SCHEMBL8097497 0.87 GPR119 (0.42) GPR119CYP11B1CYP11B2JAK2JAK1
SCHEMBL8103721 0.86 ITGB3 (0.39) KMT2AGPBAR1ERG
SCHEMBL8104346 0.85 HPGD (0.43) ALDH1A1KMT2ATSHR
SCHEMBL8088397 0.85 GAA (0.39) MEN1ALDH1A1KMT2AGPBAR1L3MBTL1
SCHEMBL8095919 0.85 ALOX12 (0.40) KMT2AGPBAR1L3MBTL1ERG
SCHEMBL8097865 0.84 L3MBTL1 (0.46) MEN1ALDH1A1MAPTKMT2AL3MBTL1
SCHEMBL8097401 0.84 GPR119 (0.43) GPR119MEN1ALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127366-A ANTICARCINOGENIC OR ANTITUMOR AGENTS MERCK & CO., INC. (US) 2000-10-03 US disclosed
US-5817678-A IMIDAZOLE-CONTAINING PIPERIDINE DERIVATIVES, PEPTIDEMIMETIC MERCK & CO., INC. (US) 1998-10-06 US disclosed