SCHEMBL8097714

SCHEMBL8097714

Nc1cc(C2(S(=O)(=O)c3ccccn3)CC2)nc(-c2ccc(NC(=O)NCC(F)F)cc2)n1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.39
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
PIK3CD O00329 4/20 0.36
NPC1 O15118 3/20 0.36
ATR Q13535 1/20 0.36
RAB9A P51151 2/20 0.35
KMT2A Q03164 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALOX15 P16050 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
GLA P06280 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
IGF1R P08069 1/20 0.34
PIK3CA P42336 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8098769 0.92 NAMPT (0.39) NAMPTCA12CA1CA2CA9
SCHEMBL8099965 0.88 NAMPT (0.39) NAMPTCA12CA1CA2CA9
SCHEMBL8091924 0.88 NAMPT (0.39) NAMPTCA12CA1CA2CA9
SCHEMBL8096070 0.86 MTOR (0.40) NAMPTPIK3CDATRKMT2AIGF1R
SCHEMBL8091502 0.86 NAMPT (0.39) NAMPTPIK3CDMAPTPIK3CA
SCHEMBL8092294 0.86 ROCK2 (0.39) NAMPTCA12CA1CA2CA9
SCHEMBL8092270 0.85 NPC1 (0.43) NPC1ATRRAB9AKMT2ASMN1; SMN2
SCHEMBL8098808 0.85 NAMPT (0.39) NAMPTCA12CA1CA2CA9
SCHEMBL8083970 0.85 NAMPT (0.39) NAMPTCA12CA1CA2CA9
SCHEMBL8090849 0.85 NAMPT (0.39) NAMPTCA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed