SCHEMBL8096070

SCHEMBL8096070

CNC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4ccccn4)CC3)n2)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MTOR P42345 8/20 0.40
PIK3CA P42336 6/20 0.40
PIK3CG P48736 4/20 0.40
PIK3CD O00329 3/20 0.40
ATR Q13535 1/20 0.38
NAMPT P43490 1/20 0.36
CDK1 P06493 2/20 0.36
CDK2 P24941 2/20 0.36
PIP4K2A P48426 1/20 0.35
PIP4K2B P78356 1/20 0.35
IGF1R P08069 1/20 0.35
AKT1 P31749 2/20 0.35
AKT2 P31751 2/20 0.35
KMT2A Q03164 1/20 0.34
MAOA P21397 1/20 0.34
PIK3R1 P27986 1/20 0.34
SMG1 Q96Q15 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8098135 0.96 MTOR (0.39) MTORPIK3CAPIK3CGPIK3CDATR
SCHEMBL8092294 0.90 ROCK2 (0.39) MTORPIK3CAPIK3CDATRNAMPT
SCHEMBL8092270 0.90 NPC1 (0.43) MTORPIK3CAATRKMT2APIK3R1
SCHEMBL8096681 0.90 ATR (0.40) MTORPIK3CAATRNAMPTIGF1R
SCHEMBL8091924 0.89 NAMPT (0.39) PIK3CAPIK3CDATRNAMPT
SCHEMBL8098769 0.88 NAMPT (0.39) PIK3CDATRNAMPT
SCHEMBL8098805 0.87 PIK3CD (0.36) PIK3CAPIK3CDATRNAMPTIGF1R
SCHEMBL8091129 0.87 KDR (0.40) ATR
SCHEMBL8090246 0.87 PIK3CA (0.42) MTORPIK3CAPIK3CGPIK3CDNAMPT
SCHEMBL8097714 0.86 NAMPT (0.39) PIK3CAPIK3CDATRNAMPTIGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed