Bromide

Bromide

SCHEMBL8098518

Br.CN1C2C=C(c3cc4c(Cl)cccc4s3)CC1CC2

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 known ✓ P23975 5/20 0.48
SLC6A4 known ✓ P31645 5/20 0.48
SLC6A3 known ✓ Q01959 5/20 0.48
HTR6 P50406 1/20 0.43
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
ALOX5 P09917 1/20 0.33
CHRNA7 P36544 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC9 Q9UKV0 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3542111 0.80 SLC6A2 (0.49) SLC6A2SLC6A4SLC6A3HTR6NOS3
SCHEMBL3542115 0.80 SLC6A2 (0.49) SLC6A2SLC6A4SLC6A3HTR6NOS3
SCHEMBL3062717 0.79 SLC6A4 (0.53) SLC6A2SLC6A4SLC6A3HTR6NOS3
Hydrochloric Acid SCHEMBL6498978 0.78 SLC6A4 (0.52) SLC6A2SLC6A4SLC6A3HTR6NOS3
SCHEMBL8108438 0.76 HTR6 (0.50) SLC6A2SLC6A4SLC6A3HTR6NOS3
SCHEMBL6500944 0.74 SLC6A2 (0.47) SLC6A2SLC6A4SLC6A3HTR6NOS3
SCHEMBL1021448 0.72 SLC6A2 (0.62) SLC6A2SLC6A4SLC6A3HTR6NOS3
SCHEMBL1021447 0.72 SLC6A2 (0.62) SLC6A2SLC6A4SLC6A3HTR6NOS3
Cadaverine Tartrate SCHEMBL3542909 0.72 SLC6A3 (0.48) SLC6A2SLC6A4SLC6A3HTR6MEN1
SCHEMBL1020817 0.72 SLC6A2 (0.69) SLC6A2SLC6A4SLC6A3HTR6NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6107307-A PSYCHOLOGICAL DISORDERS ELI LILLY AND COMPANY (US) 2000-08-22 US disclosed
EP-0969005-A1 Azabicyclic inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 2000-01-05 EP disclosed
WO-1999065492-A1 INHIBITION OF SEROTONIN REUPTAKE ELI LILLY AND COMPANY (US) 1999-12-23 WO disclosed