SCHEMBL8098826

SCHEMBL8098826

COc1cccc(C(=O)CCC(N)=O)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.65
CTNNB1 P35222 3/20 0.60
WNT3A P56704 3/20 0.60
CES2 O00748 1/20 0.59
CES1 P23141 1/20 0.59
PRSS1 P07477 1/20 0.56
PRSS2 P07478 1/20 0.56
PRSS3 P35030 1/20 0.56
HSD11B1 P28845 2/20 0.54
CHRM2 P08172 1/20 0.54
CHRM1 P11229 1/20 0.54
CHRM3 P20309 1/20 0.54
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
POLB P06746 1/20 0.52
BLM P54132 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
ALDH1A1 P00352 2/20 0.52
MAPT P10636 1/20 0.52
TDP1 Q9NUW8 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8269548 0.87 HSD11B1 (0.64) PARP1CTNNB1WNT3ACES2CES1
SCHEMBL30416831 0.85 ALDH1A1 (0.69) PARP1CTNNB1WNT3ACES2CES1
SCHEMBL4722288 0.85 ALDH1A1 (0.69) PARP1CTNNB1WNT3ACES2CES1
SCHEMBL3846484 0.85 PARP1 (0.67) PARP1CES2CES1PRSS1PRSS2
SCHEMBL15988793 0.84 CTNNB1 (0.74) PARP1CTNNB1WNT3ACES2CES1
SCHEMBL30416977 0.84 CTNNB1 (0.60) PARP1CTNNB1WNT3ACES2CES1
SCHEMBL3588375 0.84 CTNNB1 (0.60) PARP1CTNNB1WNT3ACES2CES1
Hydrochloric Acid SCHEMBL3849047 0.84 PARP1 (0.65) PARP1CTNNB1WNT3ACES2CES1
SCHEMBL4637827 0.83 CES2 (0.62) PARP1CTNNB1WNT3ACES2CES1
SCHEMBL19984838 0.83 CES2 (0.62) PARP1CTNNB1WNT3ACES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6051577-A TYROSINE INHIBITORS; BONE DISORDERS NOVARTIS AG (CH) 2000-04-18 US disclosed
WO-1997028161-A1 NOVEL PYRROLO[2,3-D]PYRIMIDINES AND THEIR USE AS TYROSINE KINASE INHIBITORS NOVARTIS AG (CH) 1997-08-07 WO disclosed