SCHEMBL8099545

SCHEMBL8099545

CC(C(=O)O)c1ccc(Oc2ccc(Cl)cc2Cl)c(NS(C)(=O)=O)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 4/20 0.56
PTGS2 P35354 4/20 0.54
PTGS1 P23219 3/20 0.54
PTGDR Q13258 5/20 0.52
PTGDR2 Q9Y5Y4 5/20 0.52
FFAR1 O14842 1/20 0.46
TTR P02766 2/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CCR4 P51679 1/20 0.41
CCR5 P51681 1/20 0.41
KCNH2 Q12809 1/20 0.41
MEN1 O00255 1/20 0.40
ABCC4 O15439 1/20 0.40
C5 P01031 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8481365 0.90 PTGS1 (0.53) CCR2PTGS2PTGS1PTGDRPTGDR2
SCHEMBL8092076 0.79 PTGS1 (0.47) CCR2PTGS2PTGS1PTGDRPTGDR2
SCHEMBL8104951 0.78 HPGD (0.53) PTGS2PTGS1FFAR1TTRCYP1A2
SCHEMBL15456906 0.78 CHRM1 (0.48) PTGS1
SCHEMBL8099718 0.76 PTGS1 (0.68) CCR2PTGS2PTGS1MEN1MAPT
SCHEMBL7160901 0.76 FFAR1 (0.60) CCR2PTGS2PTGS1PTGDRPTGDR2
SCHEMBL8523577 0.76 PTGS1 (0.58) CCR2PTGS2PTGS1PTGDRPTGDR2
SCHEMBL7162523 0.75 PTGS1 (0.59) CCR2PTGS2PTGS1PTGDRPTGDR2
SCHEMBL8481368 0.73 PTGS1 (0.52) CCR2PTGS2PTGS1PTGDRPTGDR2
SCHEMBL9657574 0.73 PTGS1 (0.60) CCR2PTGS2PTGS1PTGDRPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848703-B1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 2000-09-27 EP disclosed