SCHEMBL8100511

SCHEMBL8100511

CNC(=O)[C@@H](Cc1ccccc1)N(C)C(=O)[C@H](N)Cc1ccc2ccccc2c1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MC4R P32245 8/20 0.50
MC3R P41968 8/20 0.50
MC5R P33032 2/20 0.50
FCER2 P06734 2/20 0.48
GHSR Q92847 2/20 0.47
MC1R Q01726 6/20 0.45
MMP9 P14780 1/20 0.44
MMP8 P22894 1/20 0.44
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43
OPRD1 P41143 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4426088 0.87 FCER2 (0.53) FCER2GHSRMMP9MMP8
SCHEMBL4427112 0.87 FCER2 (0.53) FCER2GHSRMMP9MMP8
SCHEMBL6317992 0.87 FCER2 (0.53) FCER2GHSRMMP9MMP8
SCHEMBL8174004 0.84 MC4R (0.58) MC4RMC3RMC5RMC1R
SCHEMBL7061723 0.82 GHSR (0.47) MC4RMC3RFCER2GHSRMC1R
SCHEMBL4428281 0.81 GHSR (0.49) FCER2GHSRMMP9MMP8
SCHEMBL7368069 0.81 GHSR (0.49) FCER2GHSRMMP9MMP8
SCHEMBL7895834 0.81 MMP2 (0.50)
SCHEMBL7404019 0.81 MMP2 (0.50)
SCHEMBL6318200 0.81 GHSR (0.42) MC4RMC3RFCER2GHSRMC1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1060190-A1 NEW SALT FORMS OF (2E)- 5-AMINO-5- METHYLHEX-2- ENOIC ACID N-METHYL-N-((1R)-1-(N- METHYL-N-((1R)-1-(METHYLCARBAMOYL)-2- PHENYLETHYL)CARBAMOYL)-2- (2-NAPHTYL)ETHYL)AMIDE NOVO NORDISK A/S (DK) 2000-12-20 EP claimed
WO-1999045029-A1 NEW SALT FORMS OF (2E)- 5-AMINO-5- METHYLHEX-2- ENOIC ACID N-METHYL-N-((1R)-1-(N- METHYL-N-((1R)-1-(METHYLCARBAMOYL)-2- PHENYLETHYL)CARBAMOYL)-2- (2-NAPHTYL)ETHYL)AMIDE NOVO NORDISK A/S (DK) 1999-09-10 WO claimed