SCHEMBL8101752

SCHEMBL8101752

CCOC(=O)Cn1c(COc2ccc(C#N)cc2)nc2c(NS(=O)(=O)c3ccccc3)cccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLO1 Q04760 2/20 0.43
AR P10275 1/20 0.42
KDM4E B2RXH2 3/20 0.42
TDP1 Q9NUW8 2/20 0.42
LMNA P02545 2/20 0.42
HTT P42858 2/20 0.42
NPC1 O15118 1/20 0.42
GAA P10253 1/20 0.42
NPY1R P25929 2/20 0.42
TSHR P16473 2/20 0.41
KMT2A Q03164 1/20 0.41
SLC40A1 Q9NP59 2/20 0.39
STAT3 P40763 1/20 0.39
CACNA1H O95180 1/20 0.39
CACNA1B Q00975 1/20 0.39
BRPF1 P55201 1/20 0.39
ALDH1A1 P00352 4/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 1/20 0.38
SAE1 Q9UBE0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8029746 0.89 GLO1 (0.41) GLO1KDM4ETDP1LMNAHTT
SCHEMBL6635871 0.83 BRPF1 (0.48) ARLMNAHTTNPC1GAA
SCHEMBL6635525 0.83 AR (0.48) ARLMNAHTTGAAKMT2A
SCHEMBL8026525 0.82 ALDH1A1 (0.41) GLO1KDM4ETSHRKMT2ASLC40A1
SCHEMBL8028284 0.82 GLO1 (0.40) GLO1KDM4EGAATSHRKMT2A
SCHEMBL8026444 0.78 GLO1 (0.46) GLO1TDP1SLC40A1
SCHEMBL8026558 0.77 GLO1 (0.48) GLO1TDP1SLC40A1STAT3BRPF1
SCHEMBL8017545 0.74 F2 (0.48) GLO1TDP1LMNAKMT2ASLC40A1
SCHEMBL6642117 0.73 F2 (0.47) HTTNPC1GAAKMT2AALDH1A1
SCHEMBL8029744 0.73 F2 (0.60) LMNABRPF1ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6121308-A INDOLE AND BENZIMIDAZOLE ANTITHROMBOTIC COMPOUNDS, SUCH AS 1-METHYL-2-(N-(4-AMIDINOPHENYL)-AMINOMETHYL)-5-(N-(HYDROXYCARBONYLMETHYL) -QUINOLINE-8-SULPHONYLAMINO)-INDOLE BOEHRINGER INGELHEIM KG (DE) 2000-09-19 US disclosed