SCHEMBL8102963

SCHEMBL8102963

Clc1ccc2nc(Cl)c3nccn3c2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CUL4A Q13619 1/20 0.51
ALDH1A1 P00352 2/20 0.50
KDM4E B2RXH2 2/20 0.50
GAA P10253 2/20 0.50
GLA P06280 1/20 0.50
POLB P06746 1/20 0.50
HPGD P15428 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
HSD17B10 Q99714 1/20 0.50
PTPN1 P18031 1/20 0.48
IKBKB O14920 1/20 0.47
PDE2A O00408 2/20 0.39
PDE10A Q9Y233 2/20 0.39
MAP3K14 Q99558 2/20 0.39
MAPK8 P45983 1/20 0.39
HRH4 Q9H3N8 3/20 0.39
HRH3 Q9Y5N1 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 1/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL121472 0.84 HTR3E (0.45) CUL4AALDH1A1KDM4EHPGDIKBKB
SCHEMBL13077027 0.84 IKBKB (0.66) ALDH1A1KDM4EGAAPOLBPTPN1
SCHEMBL25824093 0.84 IKBKB (0.45) CUL4AALDH1A1KDM4EGAAGLA
SCHEMBL30973203 0.84 IKBKB (0.45) CUL4AALDH1A1KDM4EGAAGLA
SCHEMBL24832295 0.84 IKBKB (0.45) CUL4AALDH1A1KDM4EGAAGLA
SCHEMBL17895298 0.81 IKBKB (0.42) IKBKBPDE2APDE10ACYP1A2CYP2C9
SCHEMBL8118650 0.80 GRIN2D (0.49) ALDH1A1KDM4EGAAGLAPOLB
SCHEMBL120846 0.80 MAPK8 (0.54) ALDH1A1KDM4EGAAGLAHPGD
SCHEMBL30578099 0.80 MAPK8 (0.54) ALDH1A1KDM4EGAAGLAHPGD
SCHEMBL119071 0.77 HTR3E (0.39) ALDH1A1KDM4EPOLBHPGDIKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6124287-A TREATING DEPRESSION BIOMEDICA FOSCAMA INDUSTRIA CHIMICOFARMACEUTICA S.P.A. (IT) 2000-09-26 US disclosed
EP-0865442-B1 IMIDAZO[1,2-a]QUINOXALIN-4-AMINES ACTIVE AS ADENOSINE ANTAGONISTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THEREOF FOSCAMA BIOMED CHIM FARMA (IT) 2000-07-05 EP disclosed