SCHEMBL8103552

SCHEMBL8103552

CC(=O)c1ccc(-c2ccccc2)cc1Br.COc1ccc(C(C)=O)c(Br)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.51
ALDH1A1 P00352 2/20 0.51
MAPK1 P28482 2/20 0.51
CYP3A4 P08684 2/20 0.51
LMNA P02545 3/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
MAPT P10636 1/20 0.47
PKM P14618 1/20 0.47
AVPR2 P30518 1/20 0.47
GPR27 Q9NS67 1/20 0.47
ADORA3 P0DMS8 2/20 0.47
TRPV1 Q8NER1 1/20 0.47
POLB P06746 1/20 0.46
CYP1A2 P05177 2/20 0.46
PGR P06401 2/20 0.46
SLC6A2 P23975 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP2D6 P10635 1/20 0.46
PDE4A P27815 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1483201 0.89 MAPT (0.52) LMNAMAPTHTTHDAC3HDAC1
SCHEMBL30601548 0.86 ALDH1A1 (0.67) HPGDALDH1A1MAPK1CYP3A4LMNA
SCHEMBL898467 0.86 ALDH1A1 (0.67) HPGDALDH1A1MAPK1CYP3A4LMNA
SCHEMBL27542071 0.81 BACE1 (0.56) HPGDALDH1A1MAPK1CYP3A4MEN1
SCHEMBL22319299 0.78 ALDH1A1 (0.57) HPGDALDH1A1MAPK1CYP3A4LMNA
SCHEMBL11308149 0.76 CHEK1 (0.59) HPGDALDH1A1LMNAMAPTPDE4A
SCHEMBL19968665 0.76 MAPT (0.52) LMNAMAPTHDAC3HDAC1HSD11B1
Acetophenone SCHEMBL1481981 0.76 MAPT (0.58) LMNAMAPTHDAC8SMN1; SMN2AKR1C3
SCHEMBL27918808 0.76 ACMSD (0.63) AKR1C3AKR1C2
SCHEMBL1180221 0.76 LCK (0.58) HPGDALDH1A1MAPK1CYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973936-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 2000-01-26 EP disclosed
WO-1998046786-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed