SCHEMBL8104528

SCHEMBL8104528

CS(=O)(=O)c1ccc(C(=C2CCC2)c2ccccc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.54
SETD7 Q8WTS6 1/20 0.46
LMNA P02545 1/20 0.46
CHRM2 P08172 1/20 0.46
CYP2D6 P10635 1/20 0.46
CHRM1 P11229 1/20 0.46
CHRM3 P20309 1/20 0.46
HTR2A P28223 1/20 0.46
HRH1 P35367 1/20 0.46
HTR2B P41595 1/20 0.46
CHRNA4 P43681 1/20 0.46
HTR3A P46098 1/20 0.46
KCNH2 Q12809 1/20 0.46
ESR2 Q92731 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8103928 0.97 PTGS2 (0.54) PTGS2SETD7LMNACHRM2CYP2D6
SCHEMBL5698447 0.85 PTGS2 (0.59) PTGS2ESR2
SCHEMBL22773331 0.82 SETD7 (0.50) PTGS2SETD7LMNA
SCHEMBL8397422 0.82 PTGS2 (0.55) PTGS2ESR2
SCHEMBL8112035 0.81 PTGS2 (0.49) PTGS2
SCHEMBL8112034 0.81 PTGS2 (0.49) PTGS2
SCHEMBL22491507 0.75 GPR119 (0.53)
SCHEMBL8394302 0.75 ALDH1A1 (0.42) PTGS2CHRM2CHRM1
SCHEMBL6583952 0.74 PTGS2 (0.65) PTGS2
SCHEMBL10226596 0.74 PTGS2 (0.65) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0971910-A1 ALPHA-METHYLENE GAMMA LACTONES AS SELECTIVE CYCLOOXYGENASE-2 INHIBITORS Merck Frosst Canada & Co. (CA) 2000-01-19 EP claimed
WO-1998043966-A1 ALPHA-METHYLENE GAMMA LACTONES AS SELECTIVE CYCLOOXYGENASE-2 INHIBITORS MERCK FROSST CANADA & CO. (CA) 1998-10-08 WO claimed
EP-0971910-A1 ALPHA-METHYLENE GAMMA LACTONES AS SELECTIVE CYCLOOXYGENASE-2 INHIBITORS Merck Frosst Canada & Co. (CA) 2000-01-19 EP disclosed
WO-1998043966-A1 ALPHA-METHYLENE GAMMA LACTONES AS SELECTIVE CYCLOOXYGENASE-2 INHIBITORS MERCK FROSST CANADA & CO. (CA) 1998-10-08 WO disclosed