SCHEMBL8104707

SCHEMBL8104707

CC(C)Oc1ccc(NC(=O)CN(C)c2cccc(C#N)c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.47
ALDH1A1 P00352 6/20 0.46
MAPT P10636 3/20 0.46
HTT P42858 1/20 0.46
PSMB5 P28074 1/20 0.45
LMNA P02545 3/20 0.45
KMT2A Q03164 2/20 0.45
TP53 P04637 2/20 0.45
NLRP1 Q9C000 1/20 0.45
KDM4E B2RXH2 1/20 0.45
MCL1 Q07820 1/20 0.45
HSD17B10 Q99714 1/20 0.45
GLA P06280 1/20 0.42
GAA P10253 2/20 0.42
MAPK14 Q16539 1/20 0.42
SMO Q99835 1/20 0.42
MAPK1 P28482 1/20 0.41
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.40
MAOB P27338 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8113537 0.86 ALDH1A1 (0.48) MCHR1ALDH1A1MAPTHTTLMNA
SCHEMBL8104603 0.85 MCHR1 (0.46) MCHR1ALDH1A1MAPTHTTPSMB5
SCHEMBL8119058 0.84 MCHR1 (0.45) MCHR1ALDH1A1MAPTHTTPSMB5
SCHEMBL8113921 0.84 RORC (0.46) MCHR1ALDH1A1MAPTPSMB5LMNA
SCHEMBL8112799 0.83 PSMB5 (0.47) MCHR1ALDH1A1MAPTHTTPSMB5
SCHEMBL8114583 0.83 MCHR1 (0.44) MCHR1ALDH1A1MAPTHTTPSMB5
SCHEMBL8115072 0.80 PLAU (0.43) MCHR1ALDH1A1MAPTHTTPSMB5
Hydrochloric Acid SCHEMBL8120596 0.79 PRSS1 (0.48) ALDH1A1MAPTLMNAKMT2ATP53
SCHEMBL8119981 0.79 ALDH1A1 (0.62) MCHR1ALDH1A1MAPTLMNAKMT2A
SCHEMBL8118516 0.78 GPR34 (0.47) ALDH1A1MAPTHTTPSMB5LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1020434-A1 3-AMIDINOANILINE DERIVATIVES, ACTIVATED BLOOD COAGULATION FACTOR X INHIBITORS, AND INTERMEDIATES FOR PRODUCING BOTH Kissei Pharmaceutical Co., Ltd. (JP) 2000-07-19 EP disclosed