SCHEMBL8105044

SCHEMBL8105044

Nc1ccc(S(N)(=O)=O)cc1Sc1ccc(Br)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 13/20 0.54
CA9 Q16790 11/20 0.54
CA1 P00915 10/20 0.54
CA12 O43570 8/20 0.54
CA7 P43166 7/20 0.54
CA4 P22748 7/20 0.54
CA6 P23280 4/20 0.54
CA5A P35218 4/20 0.54
CA14 Q9ULX7 4/20 0.54
CA5B Q9Y2D0 4/20 0.54
ALDH1A1 P00352 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
HPGD P15428 1/20 0.47
CYP2C19 P33261 1/20 0.47
HSD17B10 Q99714 1/20 0.47
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8107832 0.84 CA12 (0.53) CA2CA9CA1CA12CA7
SCHEMBL8105269 0.81 PTGS2 (0.48) CA2CA9CA1CA12CA7
SCHEMBL8105352 0.80 CA2 (0.51) CA2CA9CA1CA12CA5A
SCHEMBL8101207 0.77 PTGS2 (0.54) CA2CA9CA1CA12CA4
SCHEMBL8091331 0.75 CA1 (0.49) CA2CA9CA1CA12CA7
SCHEMBL22815435 0.73 PDE7A (0.45) ALDH1A1CYP1A2CYP2C9HPGDCYP2C19
SCHEMBL878968 0.72 CA2 (1.00) CA2CA9CA1CA12CA7
SCHEMBL30351262 0.72 CA2 (1.00) CA2CA9CA1CA12CA7
SCHEMBL183959 0.71 CA2 (1.00) CA2CA9CA1CA12CA7
SCHEMBL8099561 0.71 CA1 (0.56) CA2CA9CA1CA12CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848703-B1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 2000-09-27 EP disclosed
US-6004948-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS; SIDE EFFECT REDUCTION NYCOMED AUSTRIA GMBH (AT) 1999-12-21 US disclosed
EP-0848703-A1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II Nycomed Austria GmbH (AT) 1998-06-24 EP disclosed
WO-1997003953-A1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 1997-02-06 WO disclosed