SCHEMBL8105352

SCHEMBL8105352

NS(=O)(=O)c1ccc([N+](=O)[O-])c(Sc2ccc(Br)cc2)c1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA2 P00918 8/20 0.51
CA12 O43570 4/20 0.51
CA9 Q16790 4/20 0.51
CA1 P00915 3/20 0.51
PDE7A Q13946 5/20 0.50
VCAM1 P19320 1/20 0.47
PDE7B Q9NP56 2/20 0.43
CA5A P35218 1/20 0.41
MAPT P10636 4/20 0.40
SLC6A4 P31645 1/20 0.40
NPC1 O15118 1/20 0.40
PKM P14618 1/20 0.40
MAPK1 P28482 1/20 0.40
KMT2A Q03164 1/20 0.40
POLB P06746 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8098834 0.86 PDE7A (0.64) CA2CA12CA9CA1PDE7A
SCHEMBL8104943 0.83 CA2 (0.48) CA2CA12CA9CA1PDE7A
SCHEMBL8105044 0.80 CA2 (0.54) CA2CA12CA9CA1CA5A
SCHEMBL22815433 0.78 PDE7A (0.74) PDE7APDE7BMAPTMAPK1KMT2A
SCHEMBL8107622 0.77 IDO1 (0.55) CA2CA12CA9CA1PDE7A
SCHEMBL8107806 0.74 VCAM1 (0.56) CA2CA12CA9CA1PDE7A
SCHEMBL8101207 0.73 PTGS2 (0.54) CA2CA12CA9CA1SLC6A4
SCHEMBL29242001 0.72 CA2 (0.68) CA2CA12CA9CA1VCAM1
SCHEMBL4607929 0.72 PDE7A (0.55) PDE7APDE7BMAPTMAPK1KMT2A
SCHEMBL27915770 0.71 CA2 (0.72) CA2CA12CA9CA1VCAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848703-B1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 2000-09-27 EP disclosed
US-6004948-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS; SIDE EFFECT REDUCTION NYCOMED AUSTRIA GMBH (AT) 1999-12-21 US disclosed
EP-0848703-A1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II Nycomed Austria GmbH (AT) 1998-06-24 EP disclosed
WO-1997003953-A1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 1997-02-06 WO disclosed