SCHEMBL8106592

SCHEMBL8106592

N#CC1(c2ccsc2)CCC1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
LMNA P02545 2/20 0.35
TP53 P04637 1/20 0.35
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
OPRM1 P35372 4/20 0.35
CHRM1 P11229 1/20 0.33
WDR5 P61964 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11588203 0.96 NPC1 (0.39) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL11591376 0.94 ALDH1A1 (0.38) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL4446561 0.92 OPRM1 (0.37) OPRM1CHRM1
SCHEMBL14294295 0.83 CHRM1 (0.37) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL4767078 0.82 PDE4A (0.41) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL6337276 0.80 NPC1 (0.31) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL4762122 0.79 OPRM1 (0.30) OPRM1
SCHEMBL14258204 0.77 KMT2A (0.33) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL8317825 0.74 KCNA3 (0.37) CHRM1
SCHEMBL872608 0.72 OPRM1 (0.56) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116987095-A Spiro-containing derivative, preparation method and application thereof 上海枢境生物科技有限公司 2023-11-03 CN disclosed
CN-116057060-B Spiro-containing derivative, preparation method and application thereof 上海枢境生物科技有限公司 2023-08-29 CN disclosed
CN-116057060-A Spiro-containing derivative, preparation method and application thereof 上海枢境生物科技有限公司 2023-05-02 CN disclosed
WO-2022206706-A1 SPIRO-CONTAINING DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海枢境生物科技有限公司 2022-10-06 WO disclosed
US-6124354-A TREATMENT OF URINARY INCONTINENCE OR IRRITABLE BOWEL SYNDROME PHARMACIA & UPJOHN AB (SE) 2000-09-26 US disclosed