SCHEMBL8107574

SCHEMBL8107574

CN(C)CC[C@@H](O)[C@@H]1C[C@H](SC(c2ccccc2)(c2ccccc2)c2ccccc2)CN1C(=O)OCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 6/20 0.42
TDP1 Q9NUW8 1/20 0.39
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8112388 0.90 CCR5 (0.39) CCR5TDP1ATM
SCHEMBL8112453 0.89 CCR5 (0.38) CCR5
SCHEMBL9569904 0.88 TDP1 (0.43) CCR5TDP1ATM
SCHEMBL9137735 0.87 CCR5 (0.43) CCR5TDP1ATM
SCHEMBL7860693 0.81 TDP1 (0.43) CCR5TDP1ATM
SCHEMBL7805543 0.81 TDP1 (0.43) CCR5TDP1ATM
SCHEMBL7811582 0.81 TDP1 (0.43) CCR5TDP1ATM
SCHEMBL9519179 0.81 TDP1 (0.42) CCR5TDP1ATM
SCHEMBL9265469 0.81 DPP4 (0.43) CCR5TDP1ATM
SCHEMBL9521184 0.81 TDP1 (0.42) CCR5TDP1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0545290-B1 Aminoalkylpyrrolidinylthiocarbapenem derivatives BANYU PHARMA CO LTD (JP) 2000-08-23 EP disclosed
US-5550121-A ANTIBIOTICS BANYU PHARMACEUTICAL CO., LTD. (JP) 1996-08-27 US disclosed
EP-0545290-A1 Aminoalkylpyrrolidinylthiocarbapenem derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-06-09 EP disclosed