SCHEMBL8108170

SCHEMBL8108170

O=c1cc(-c2ccc(F)cc2)nc2ccc(Cl)cn12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSD A5PKW4 2/20 0.48
MAPT P10636 2/20 0.46
TP53 P04637 2/20 0.46
THRB P10828 1/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
KDM5B Q9UGL1 2/20 0.44
SIRT5 Q9NXA8 1/20 0.44
RAD51 Q06609 1/20 0.43
CDC7 O00311 1/20 0.43
PIM1 P11309 1/20 0.43
GSK3B P49841 1/20 0.43
HIPK2 Q9H2X6 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
NTRK1 P04629 1/20 0.42
NTRK2 Q16620 1/20 0.42
DHODH Q02127 1/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CRHBP P24387 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28958142 0.85 NPC1 (0.56) MAPTNPC1RAB9ARAD51MEN1
SCHEMBL8092460 0.83 GRIN1 (0.55) MAPTTP53THRBNPC1RAB9A
SCHEMBL8106156 0.81 PKM (0.45) MAPTNPC1RAB9AMEN1ALDH1A1
SCHEMBL8099805 0.80 NPC1 (0.58) MAPTTP53NPC1RAB9ARAD51
SCHEMBL15175242 0.77 ALDH1A3 (0.48) MAPTTP53NPC1RAB9APKM
SCHEMBL8092386 0.77 NPC1 (0.55) MAPTTP53THRBNPC1RAB9A
SCHEMBL15175532 0.75 ENPP2 (0.51) MAPTTP53THRBKDM5BRAD51
SCHEMBL13325716 0.74 RAB9A (0.81) MAPTNPC1RAB9AMEN1ALDH1A1
SCHEMBL15175573 0.74 FYN (0.39) MAPTTP53THRBKDM5B
SCHEMBL31314523 0.74 FYN (0.39) MAPTTP53THRBKDM5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6071930-A FOR INHIBITION OF MITOSIS OR TUMOR GROWTH THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2000-06-06 US disclosed