SCHEMBL8109302

SCHEMBL8109302

CC(=O)N(C)c1c(C(=O)OC(C)C(=O)c2cc(Cl)ccn2)[nH]c2cc(Cl)ccc12

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 6/20 0.38
MDM2 Q00987 3/20 0.37
KDM4C Q9H3R0 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
GSK3B P49841 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8116085 0.83 ALOX15 (0.41) ALOX15KDM4CALDH1A1MAPTGSK3B
SCHEMBL7501925 0.83 PTGS2 (0.44) ALOX15ALDH1A1MAPTL3MBTL1GSK3B
SCHEMBL6171070 0.76 PTGS2 (0.48) ALOX15
SCHEMBL6171153 0.69 TUBB4A (0.44) ALOX15MDM2
SCHEMBL7506944 0.69 GSK3B (0.40) ALOX15KDM4CALDH1A1GSK3B
SCHEMBL7507324 0.68 ALOX15 (0.40) ALOX15ALDH1A1MAPT
SCHEMBL8137033 0.67 ABCB11 (0.46) ALOX15GSK3B
SCHEMBL8117061 0.67 ALOX15 (0.41) ALOX15MDM2ALDH1A1MAPTL3MBTL1
SCHEMBL6170606 0.66 PTGS2 (0.48) MDM2KDM4CMAPT
SCHEMBL7502692 0.66 MEN1 (0.46) ALOX15MDM2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001934-A1 INDOLE COMPOUNDS AS COX-2 INHIBITORS PFIZER PHARMACEUTICALS INC. (JP) 2000-05-24 EP disclosed
WO-1999005104-A1 INDOLE COMPOUNDS AS COX-2 INHIBITORS PFIZER PHARMACEUTICALS INC. (JP) 1999-02-04 WO disclosed