SCHEMBL8109351

SCHEMBL8109351

Cc1c(N2C(=O)c3ccccc3C2=O)c(CCl)nc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
KDM4E B2RXH2 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
KMT2A Q03164 3/20 0.46
MAPT P10636 3/20 0.40
ALPL P05186 1/20 0.39
RAB9A P51151 1/20 0.39
TSHR P16473 1/20 0.39
GAA P10253 2/20 0.39
MAPK1 P28482 2/20 0.38
POLB P06746 1/20 0.38
MEN1 O00255 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CASP3 P42574 1/20 0.38
CYP1A2 P05177 1/20 0.37
GLA P06280 1/20 0.37
CYP3A4 P08684 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1721513 0.82 KMT2A (0.42) ALDH1A1KDM4ESMN1; SMN2KMT2AMAPT
SCHEMBL1722353 0.76 PDE7A (0.43) ALDH1A1KDM4ESMN1; SMN2KMT2AMAPT
SCHEMBL8109356 0.76 GRM5 (0.43) KDM4ESMN1; SMN2KMT2AMAPTRAB9A
SCHEMBL12204686 0.68 KMT2A (0.53) ALDH1A1KMT2ATSHRGAAPOLB
SCHEMBL9837203 0.68 RXFP1 (0.38) ALDH1A1KMT2AMAPTALPLGAA
SCHEMBL3971941 0.67 KMT2A (0.53) ALDH1A1KDM4ESMN1; SMN2KMT2AMAPT
SCHEMBL18470455 0.65 KMT2A (1.00) ALDH1A1KDM4ESMN1; SMN2KMT2AMAPT
SCHEMBL824417 0.64 RAB9A (0.65) ALDH1A1KDM4ESMN1; SMN2KMT2AMAPT
SCHEMBL13957877 0.63 DHODH (0.48) ALDH1A1KDM4EKMT2ATSHRGAA
SCHEMBL9362074 0.63 KDM4E (0.54) ALDH1A1KDM4ESMN1; SMN2KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6121308-A INDOLE AND BENZIMIDAZOLE ANTITHROMBOTIC COMPOUNDS, SUCH AS 1-METHYL-2-(N-(4-AMIDINOPHENYL)-AMINOMETHYL)-5-(N-(HYDROXYCARBONYLMETHYL) -QUINOLINE-8-SULPHONYLAMINO)-INDOLE BOEHRINGER INGELHEIM KG (DE) 2000-09-19 US disclosed