SCHEMBL8109356

SCHEMBL8109356

Cc1c(N2C(=O)c3ccccc3C2=O)c(COc2ccc(C#N)cc2)nc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.43
LMNA P02545 1/20 0.42
PKM P14618 1/20 0.42
MAPK1 P28482 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
MAOB P27338 2/20 0.40
PDCD1 Q15116 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ATM Q13315 1/20 0.40
AR P10275 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
RAB9A P51151 1/20 0.38
GBA1 P04062 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8109351 0.76 ALDH1A1 (0.47) MAPK1SMN1; SMN2MEN1KMT2AKDM4E
SCHEMBL6785535 0.72 NPC1 (0.53) LMNAMAPK1SMN1; SMN2RXFP1MAOB
SCHEMBL6635377 0.72 PDCD1 (0.42) GRM5PKMMAPK1SMN1; SMN2RXFP1
SCHEMBL6638692 0.71 GRM5 (0.48) GRM5MAOBPDCD1CD274MEN1
SCHEMBL1721513 0.69 KMT2A (0.42) LMNAMAPK1SMN1; SMN2MEN1KMT2A
SCHEMBL1722353 0.67 PDE7A (0.43) MAPK1SMN1; SMN2RXFP1MEN1KMT2A
SCHEMBL30010206 0.66 PDCD1 (0.70) GRM5PDCD1CD274
SCHEMBL28590561 0.66 PDCD1 (0.70) GRM5PDCD1CD274
SCHEMBL13107075 0.65 SMN1; SMN2 (0.42) PKMMAPK1SMN1; SMN2RXFP1MAOB
SCHEMBL13096745 0.64 MAOB (0.48) LMNAPKMMAPK1SMN1; SMN2RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6121308-A INDOLE AND BENZIMIDAZOLE ANTITHROMBOTIC COMPOUNDS, SUCH AS 1-METHYL-2-(N-(4-AMIDINOPHENYL)-AMINOMETHYL)-5-(N-(HYDROXYCARBONYLMETHYL) -QUINOLINE-8-SULPHONYLAMINO)-INDOLE BOEHRINGER INGELHEIM KG (DE) 2000-09-19 US disclosed