SCHEMBL8109897

SCHEMBL8109897

CCC(C(=O)O)C(NC(=O)CC1CCN(c2ccc(C=NN)cc2)C1=O)c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.36
KEAP1 Q14145 2/20 0.34
NFE2L2 Q16236 2/20 0.34
HTR1A P08908 1/20 0.33
ADRA1A P35348 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
XIAP P98170 4/20 0.32
ADAM17 P78536 2/20 0.32
DPP4 P27487 1/20 0.32
DPP8 Q6V1X1 1/20 0.32
MMP2 P08253 1/20 0.32
MMP9 P14780 1/20 0.32
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ROCK2 O75116 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8118631 0.95 CYP1A2 (0.35) PTPN1KEAP1NFE2L2HTR1AADRA1A
SCHEMBL8117806 0.88 HTT (0.31) PTPN1ADAM17HTT
SCHEMBL7532349 0.86 UGCG (0.36) KEAP1NFE2L2KMT2AADAM17LMNA
SCHEMBL8122599 0.86
SCHEMBL8122271 0.86 ITGB3 (0.36) ALDH1A1
SCHEMBL9029392 0.83 OPRM1 (0.35) PTPN1ADAM17MMP2MMP9ALDH1A1
SCHEMBL8118294 0.83 ITGB3 (0.33) CYP1A2CYP2D6CYP2C9ALDH1A1HTT
SCHEMBL8125482 0.83 ITGB3 (0.33) CYP1A2CYP2D6CYP2C9ALDH1A1HTT
SCHEMBL7417886 0.83 ITGB3 (0.42) PTPN1ALDH1A1SMN1; SMN2
SCHEMBL7421979 0.82 LMNA (0.44) PTPN1KMT2AADAM17DPP4DPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691953-B1 1-AMIDINOPHENYL-PYRROLIDONES/ PIPERIDINONES AS PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 2000-08-02 EP claimed