SCHEMBL810996

SCHEMBL810996

Cc1cc(NC(=NC#N)NCCCCCCNC(=O)c2ccc(Cl)cc2)ccn1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.53
PSEN2 P49810 1/20 0.53
APH1B Q8WW43 1/20 0.53
NCSTN Q92542 1/20 0.53
APH1A Q96BI3 1/20 0.53
PSENEN Q9NZ42 1/20 0.53
RAB9A P51151 2/20 0.48
NPC1 O15118 1/20 0.48
IKBKB O14920 1/20 0.44
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL810378 0.86 IKBKB (0.56) IKBKBHDAC3HDAC4HDAC1HDAC7
SCHEMBL810725 0.79 KCNJ11 (0.54) RAB9ANPC1IKBKBHDAC3HDAC4
SCHEMBL504263 0.79 PSEN1 (0.51) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL504262 0.79 PSEN1 (0.51) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6615293 0.77 CYP11B1 (0.57) RAB9AMEN1KMT2A
SCHEMBL810930 0.76 IKBKB (0.54) RAB9ANPC1IKBKBHDAC3HDAC4
SCHEMBL811142 0.76 IKBKB (0.54) RAB9ANPC1IKBKBHDAC3HDAC4
SCHEMBL810238 0.76 IKBKB (0.54) RAB9ANPC1IKBKBHDAC3HDAC4
SCHEMBL16312363 0.75 IKBKB (0.64) RAB9ANPC1IKBKBSMARCA2SMARCA4
SCHEMBL810405 0.75 CYP1A2 (0.50) RAB9AIKBKBHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2394649-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING PYRIDYL CYANOGUANIDINES, PREPARATION METHODS AND USES THEREOF Tianjin Hemay Bio-Tech Co., Ltd. (CN) 2011-12-14 EP disclosed