SCHEMBL8110697

SCHEMBL8110697

[O-][S+]1CNc2ccc(CCCCN3CCC(Cc4ccccc4)CC3)cc21

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.60
CCR3 P51677 2/20 0.60
GRIN2B Q13224 1/20 0.53
ABCB1 P08183 1/20 0.52
HRH3 Q9Y5N1 1/20 0.50
KCNH2 Q12809 1/20 0.49
SLC6A2 P23975 2/20 0.48
SLC6A4 P31645 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8116069 0.93 CCR3 (0.57) SIGMAR1CCR3GRIN2BABCB1SLC6A2
SCHEMBL8958333 0.87 SIGMAR1 (0.58) SIGMAR1
SCHEMBL8114275 0.83 GRIN2B (0.49) CCR3GRIN2BSLC6A2SLC6A4
SCHEMBL9449426 0.83 SIGMAR1 (0.57) SIGMAR1KCNH2
SCHEMBL8110476 0.80 SIGMAR1 (0.61) SIGMAR1CCR3GRIN2BABCB1HRH3
SCHEMBL8109932 0.79 SIGMAR1 (0.47) SIGMAR1
SCHEMBL7756732 0.79 DRD2 (0.45) SIGMAR1HRH3SLC6A4
SCHEMBL7756751 0.78 SIGMAR1 (0.44) SIGMAR1HRH3KCNH2SLC6A2SLC6A4
SCHEMBL7374609 0.77 SIGMAR1 (1.00) SIGMAR1CCR3HRH3KCNH2SLC6A2
SCHEMBL7763028 0.76 SIGMAR1 (0.37) SIGMAR1HRH3SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0673933-B1 Aminoalkyl benzoxazolinones and benzothiazolinones process for their preparation and compositions containing them ADIR (FR) 2000-11-08 EP disclosed
US-5534511-A AFFINITY FOR SIGMA RECEPTORS, ANTIINFLAMMATORY, TREATMENT OF ARTHRITIS ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
EP-0673933-A1 Aminoalkyl benzoxazolinones and benzothiazolinones process for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1995-09-27 EP disclosed